SCHEMBL7783488

SCHEMBL7783488

O=c1[nH]c(-c2ccc(C(F)(F)F)cc2)nc2c1CSCC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TNKS2 Q9H2K2 15/20 1.00
TNKS O95271 11/20 1.00
WNT3A P56704 9/20 1.00
PARP1 P09874 7/20 1.00
PARP2 Q9UGN5 6/20 1.00
PARP3 Q9Y6F1 2/20 1.00
PARP14 Q460N5 1/20 1.00
PARP4 Q9UKK3 1/20 1.00
AXIN2 Q9Y2T1 1/20 1.00
BRD4 O60885 1/20 0.51
PARP15 Q460N3 1/20 0.50
COMT P21964 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30870719 0.88 TNKS2 (0.78) TNKS2TNKSWNT3APARP1PARP2
SCHEMBL30870677 0.86 TNKS2 (0.75) TNKS2TNKSWNT3APARP1PARP2
SCHEMBL27438107 0.85 TNKS2 (0.82) TNKS2TNKSWNT3APARP1PARP2
SCHEMBL27438444 0.84 TNKS2 (0.80) TNKS2TNKSWNT3APARP1PARP2
SCHEMBL7776852 0.84 TNKS2 (0.73) TNKS2TNKSWNT3APARP1PARP2
SCHEMBL7783311 0.83 TNKS2 (0.71) TNKS2TNKSWNT3APARP1PARP2
SCHEMBL7782072 0.83 TNKS2 (0.71) TNKS2TNKSWNT3APARP1PARP2
SCHEMBL27436932 0.83 TNKS2 (0.71) TNKS2TNKSWNT3APARP1PARP2
SCHEMBL7783581 0.83 TNKS2 (0.70) TNKS2TNKSWNT3APARP1PARP2
SCHEMBL27436124 0.82 TNKS2 (0.70) TNKS2TNKSWNT3APARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2082 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026106998-A1 PROSTATE-SPECIFIC MEMBRANE ANTIGEN (PSMA)-TARGETED POLY(ADP-RIBOSE) POLYMERASE (PARP) INHIBITOR AND RELATED COMPOSITION AND METHOD OF USE PURDUE RESEARCH FOUNDATION (US) 2026-05-21 WO claimed
CN-122038285-A Kit and method for constructing human bone organ by using pluripotent stem cells 广东医科大学附属医院 2026-05-15 CN claimed
WO-2025251988-A9 REAGENT COMBINATION OR KIT FOR CONSTRUCTING EMBRYOID AND USE THEREOF 广州国家实验室 2026-05-15 WO claimed
EP-4739310-A1 ECTONUCLEOTIDE PYROPHOSPHATASE/PHOSPHODIESTERASE 1 (ENPP1) INHIBITOR COMBINATIONS AND USES THEREOF Insilico Medicine IP Limited (HK) 2026-05-13 EP claimed
US-12624339-B2 Brain organoid containing optic vesicles generated based on H9 induction and eye-brain fusion culture method TIANJIN UNIVERSITY (CN) 2026-05-12 US claimed
US-20260124249-A1 USE OF TNKS INHIBITORS FOR REGENERATION OF CARTILAGE LIFLEX SCIENCE INC. (KR) 2026-05-07 US claimed
US-20260125650-A1 METHODS AND COMPOSITIONS FOR GENERATING HEPATOCYTES TRAILHEAD BIOSYSTEMS INC (US) 2026-05-07 US claimed
EP-4728051-A1 STANDARDISING PLURIPOTENT STEM CELLS United Kingdom Research and Innovation (GB) 2026-04-22 EP claimed
EP-3964565-B1 AN IN VITRO METHOD OF DIFFERENTIATING A HUMAN PLURIPOTENT STEM CELL POPULATION INTO A CARDIOMYOCYTE CELL POPULATION NCARDIA B V (NL) 2026-04-08 EP claimed
US-20260069600-A1 COMBINATION DRUG CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2026-03-12 US claimed
US-10064862-B2 Antiviral axin stabilizer THE BOARD OF REGENTS FOR OKLAHOMA STATE UNIVERSITY (US) 2018-09-04 US claimed
EP-3347456-A1 METHOD FOR REPRODUCIBLE DIFFERENTIATION OF CLINICAL-GRADE RETINAL PIGMENT EPITHELIUM CELLS The United States of America, as represented by The Secretary, Department of Health and Human Services (US) 2018-07-18 EP claimed
US-20180195046-A1 INDUCED EXTENDED PLURIPOTENT STEM CELLS, METHOD OF MAKING AND USING PEKING UNIVERSITY (CN) 2018-07-12 US claimed
EP-2951290-B1 METHOD FOR GENERATING RETINAL PIGMENT EPITHELIUM (RPE) CELLS FROM INDUCED PLURIPOTENT STEM CELLS (IPSCS) US HEALTH (US) 2017-11-29 EP claimed
WO-2017044483-A1 METHOD FOR REPRODUCIBLE DIFFERENTIATION OF CLINICAL-GRADE RETINAL PIGMENT EPITHELIUM CELLS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2017-03-16 WO claimed
US-20170065587-A1 ANTIVIRAL AXIN STABLIZER THE BOARD OF REGENTS FOR OKLAHOMA STATE UNIVERSITY 2017-03-09 US claimed
EP-2951290-A2 METHOD FOR GENERATING RETINAL PIGMENT EPITHELIUM (RPE) CELLS FROM INDUCED PLURIPOTENT STEM CELLS (IPSCs) The United States of America, as represented by The Secretary, Department of Health and Human Services (US) 2015-12-09 EP claimed
WO-2015134525-A1 ANTIVIRAL AXIN STABILIZER THE BOARD OF REGENTS FOR OKLAHOMA STATE UNIVERSITY (US) 2015-09-11 WO claimed
WO-2014121077-A2 METHOD FOR GENERATING RETINAL PIGMENT EPITHELIUM (RPE) CELLS FROM INDUCED PLURIPOTENT STEM CELLS (IPSCs) THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2014-08-07 WO claimed
US-20130273649-A1 Culture medium for pluripotent stem cells UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2013-10-17 US claimed