SCHEMBL7783700

SCHEMBL7783700

COc1cc(CN2CC(C)CCn3c(c(-c4ccccc4)c4cccnc4c3=O)C2=O)cc(OC)c1

nearest known ligand 0.67

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 8/20 0.67
PDE4A P27815 5/20 0.40
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38
TNIK Q9UKE5 2/20 0.36
WDR5 P61964 2/20 0.34
KCNH2 Q12809 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6788330 1.00 TACR1 (0.67) TACR1PDE4AROCK2ROCK1TNIK
SCHEMBL7785041 0.94 TACR1 (0.76) TACR1PDE4AROCK2ROCK1TNIK
SCHEMBL6795274 0.94 TACR1 (0.76) TACR1PDE4AROCK2ROCK1TNIK
SCHEMBL6801261 0.93 TACR1 (0.68) TACR1PDE4AROCK2ROCK1TNIK
SCHEMBL6788387 0.93 TACR1 (0.66) TACR1PDE4AROCK2ROCK1KCNH2
SCHEMBL7786545 0.93 TACR1 (0.68) TACR1PDE4AROCK2ROCK1TNIK
SCHEMBL7783707 0.90 TACR1 (0.62) TACR1PDE4AROCK2ROCK1TNIK
SCHEMBL6800012 0.90 TACR1 (0.62) TACR1PDE4AROCK2ROCK1TNIK
SCHEMBL6799323 0.88 TACR1 (0.72) TACR1PDE4AKCNH2HRH3
SCHEMBL6794855 0.86 TACR1 (0.75) TACR1PDE4AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1145714-A1 DRUGS Takeda Chemical Industries, Ltd. (JP) 2001-10-17 EP disclosed