SCHEMBL7783707

SCHEMBL7783707

COc1cc(CN2CC(C)CCn3c(c(-c4ccc(Cl)c(Cl)c4)c4cccnc4c3=O)C2=O)cc(OC)c1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 8/20 0.62
PDE4A P27815 8/20 0.37
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
TNIK Q9UKE5 1/20 0.35
ALDH1A1 P00352 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
NPC1 O15118 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6800012 1.00 TACR1 (0.62) TACR1PDE4AROCK2ROCK1TNIK
SCHEMBL6788387 0.92 TACR1 (0.66) TACR1PDE4AROCK2ROCK1
SCHEMBL6801280 0.91 TACR1 (0.52) TACR1PDE4AROCK2ROCK1TNIK
SCHEMBL6795400 0.90 TACR1 (0.51) TACR1PDE4AROCK2ROCK1TNIK
SCHEMBL6799162 0.90 TACR1 (0.69) TACR1PDE4A
SCHEMBL6795274 0.90 TACR1 (0.76) TACR1PDE4AROCK2ROCK1TNIK
SCHEMBL7785041 0.90 TACR1 (0.76) TACR1PDE4AROCK2ROCK1TNIK
SCHEMBL7783700 0.90 TACR1 (0.67) TACR1PDE4AROCK2ROCK1TNIK
SCHEMBL6788330 0.90 TACR1 (0.67) TACR1PDE4AROCK2ROCK1TNIK
SCHEMBL6801261 0.89 TACR1 (0.68) TACR1PDE4AROCK2ROCK1TNIK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1145714-A1 DRUGS Takeda Chemical Industries, Ltd. (JP) 2001-10-17 EP disclosed