SCHEMBL7784176

SCHEMBL7784176

CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=O)N1CC(=O)O

nearest known ligand 0.74

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AR P10275 6/20 0.71
PGR P06401 1/20 0.71
HDAC1 Q13547 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29757665 0.91 AR (0.70) ARPGR
SCHEMBL31581610 0.90 AR (0.79) ARPGRHDAC1
SCHEMBL4204207 0.88 AR (0.82) ARPGRHDAC1
SCHEMBL4027539 0.87 AR (0.66) ARPGR
SCHEMBL4196099 0.87 AR (0.66) ARPGR
SCHEMBL4027208 0.87 AR (0.74) ARPGR
SCHEMBL4194508 0.86 AR (0.65) ARPGR
SCHEMBL4028572 0.86 AR (0.86) ARPGR
SCHEMBL4029305 0.86 AR (0.78) ARPGR
SCHEMBL29921612 0.86 AR (0.78) ARPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0671156-B1 Process to prepare cosmetic or pharmaceutical compositions containing liposomes AVENTIS PHARMA SA (FR) 2001-10-24 EP disclosed
US-6162444-A Cosmetic or pharmaceutical compositions HOECHST MARION ROUSSEL (FR) 2000-12-19 US disclosed
US-RE35956-E Phenylimidazolidines having antiandrogenic activity ROUSSEL UCLAF (FR) 1998-11-10 US disclosed
US-5627201-A Phenylimidazolidines having antiandrogenic activity ROUSSEL UCLAF (FR) 1997-05-06 US disclosed
EP-0671156-A1 Cosmetic or pharmaceutical compositions containing liposomes ROUSSEL UCLAF (FR) 1995-09-13 EP disclosed
US-5411981-A Phenylimidazolidines having antiandrogenic activity ROUSSEL UCLAF (FR) 1995-05-02 US disclosed
EP-0580459-A1 Substituted Phenylimidazolidins, process for their preparation, their use as medicaments and their pharmaceutical compositions containing them ROUSSEL UCLAF (FR) 1994-01-26 EP disclosed