SCHEMBL7784302

SCHEMBL7784302

Nc1nc(Cl)c(C(F)(F)F)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.41
KHK P50053 1/20 0.35
BACE1 P56817 1/20 0.34
IDO1 P14902 2/20 0.33
POLB P06746 2/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
TSHR P16473 1/20 0.33
CASP3 P42574 1/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
XPO1 O14980 2/20 0.33
ADRB2 P07550 1/20 0.33
MPL P40238 1/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
SLC9A1 P19634 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31717937 1.00 PIK3CD (0.41) PIK3CDKHKBACE1IDO1POLB
SCHEMBL2947783 0.83 PIK3CD (0.41) PIK3CDKHKBACE1POLBGLA
SCHEMBL7786072 0.82 MPL (0.35) PIK3CDBACE1IDO1POLBGLA
SCHEMBL9967097 0.82 KHK (0.50) PIK3CDKHKBACE1POLBGLA
SCHEMBL29687228 0.80 PIK3CD (0.37) PIK3CDIDO1CASP3XPO1ADRB2
SCHEMBL675996 0.80 PIK3CD (0.37) PIK3CDIDO1CASP3XPO1ADRB2
SCHEMBL11276391 0.80 PIK3CD (0.39) PIK3CDKHKBACE1POLBGLA
SCHEMBL10853416 0.77 PIK3CD (0.40) PIK3CDBACE1XPO1ADRB2MPL
SCHEMBL1420767 0.77 PIK3CD (0.42) PIK3CDBACE1POLBGLAGAA
SCHEMBL21670482 0.77 NOTUM (0.35) PIK3CDIDO1CASP3HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111574439-A Method for preparing 2-amino-3 chloro-5-trifluoromethylpyridine 山东汇盟生物科技有限公司 2020-08-25 CN claimed
CN-109963851-B Fused bicyclic pyridine compounds and their use as AMPA receptor modulators 詹森药业有限公司 2021-11-30 CN disclosed
CN-111574439-A Method for preparing 2-amino-3 chloro-5-trifluoromethylpyridine 山东汇盟生物科技有限公司 2020-08-25 CN disclosed
EP-0759429-B1 Substituted trifluormethylpyridines useful as intermediates for herbicidal 1-(pyridyl)-pyrazoles BASF AG (DE) 2001-10-24 EP disclosed
EP-1140489-A1 MULTILAYER STRUCTURES THE DOW CHEMICAL COMPANY (US) 2001-10-10 EP disclosed
WO-2000024577-A1 MULTILAYER STRUCTURES THE DOW CHEMICAL COMPANY (US) 2000-05-04 WO disclosed
US-5849920-A Substituted trifluoromethylpyridines BASF AKTIENGESELLSCHAFT (DE) 1998-12-15 US disclosed
US-5750705-A HERBICIDES BASF AKTIENGESELLSCHAFT (DE) 1998-05-12 US disclosed
EP-0759429-A1 Substituted trifluormethylpyridines useful as intermediates for herbicidal 1-(pyridyl)-pyrazoles BASF Aktiengesellschaft (DE) 1997-02-26 EP disclosed
EP-0596491-B1 Method for halogenating an aromatic compound ISHIHARA SANGYO KAISHA (JP) 1996-07-10 EP disclosed
US-5491239-A Method for halogenating an aromatic compound ISHIHARA SANGYO KAISHA LTD. (JP) 1996-02-13 US disclosed
EP-0596491-A1 Method for halogenating an aromatic compound ISHIHARA SANGYO KAISHA, LTD. (JP) 1994-05-11 EP disclosed
US-4349681-A 2-Amino-3-chloro-5-trifluoromethylpyridine ISHIHARA SANGYO KAISHA, LTD. (JP) 1982-09-14 US disclosed
EP-0031218-A1 A 2-amino-trifluoromethyl-halogenopyridine compound and a process for producing the same ISHIHARA SANGYO KAISHA LTD. (JP) 1981-07-01 EP disclosed