SCHEMBL7785115

SCHEMBL7785115

O=C(Nc1ccc(NC(=S)Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1)c1cscn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.51
JUN P05412 4/20 0.49
NFKB1 P19838 4/20 0.49
NFKB2 Q00653 4/20 0.49
RELA Q04206 4/20 0.49
GRM4 Q14833 1/20 0.48
MAPT P10636 3/20 0.47
KDM4E B2RXH2 2/20 0.47
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
ALDH1A1 P00352 2/20 0.46
TEK Q02763 1/20 0.46
P2RX1 P51575 2/20 0.45
BRAF P15056 1/20 0.44
PSEN1 P49768 1/20 0.44
PSEN2 P49810 1/20 0.44
APH1B Q8WW43 1/20 0.44
NCSTN Q92542 1/20 0.44
APH1A Q96BI3 1/20 0.44
PSENEN Q9NZ42 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7905383 0.85 CYP2C9 (0.47) KDRGRM4MAPTMEN1KMT2A
SCHEMBL7743967 0.85 CYP2C9 (0.47) KDRGRM4MAPTMEN1KMT2A
SCHEMBL7908147 0.85 CYP2C9 (0.47) KDRGRM4MAPTMEN1KMT2A
SCHEMBL15701265 0.84 PSEN1 (0.50) JUNNFKB1NFKB2RELAGRM4
SCHEMBL7737922 0.83 CYP2C9 (0.44) KDRGRM4MAPTMEN1KMT2A
SCHEMBL7161969 0.83 GRM4 (0.61) KDRGRM4MEN1KMT2ATEK
SCHEMBL15701108 0.81 PSEN1 (0.57) JUNNFKB1NFKB2RELAGRM4
SCHEMBL7979004 0.81 MAPT (0.71) KDRJUNNFKB1NFKB2RELA
SCHEMBL7743480 0.80 CYP2C9 (0.44) KDRGRM4MAPTMEN1KMT2A
SCHEMBL15701038 0.79 JUN (0.46) JUNNFKB1NFKB2RELAGRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144397-A3 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING PHENYLENEDIAMINE GROUP Wyeth (US) 2002-09-11 EP disclosed
EP-1144397-A2 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-17 EP disclosed
WO-2000034258-A2 HETEROCYCLIC CARBOXAMIDE-CONTAINING THIOUREA INHIBITORS OF HERPES VIRUSES CONTAINING PHENYLENEDIAMINE GROUP AMERICAN HOME PRODUCTS CORPORATION (US) 2000-06-15 WO disclosed