SCHEMBL7786366

SCHEMBL7786366

CCOc1ccc(OC(C)C2CCCCN2)c2c1-c1c(OC(C)C3CCCCN3)cccc1C2=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.40
SLC6A2 P23975 4/20 0.39
SLC6A3 Q01959 4/20 0.39
SLC6A4 P31645 3/20 0.39
PTPRC P08575 1/20 0.38
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 1/20 0.36
APAF1 O14727 1/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
CASP1 P29466 1/20 0.36
BRCA1 P38398 1/20 0.36
CASP7 P55210 1/20 0.36
HTR2A P28223 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7786146 0.97 TTR (0.41) TTRSLC6A2SLC6A3SLC6A4PTPRC
SCHEMBL7794788 0.95 TTR (0.42) TTRSLC6A2SLC6A3SLC6A4PTPRC
SCHEMBL7792711 0.92 HTR2A (0.38) TTRSLC6A2SLC6A3SLC6A4HTR2A
SCHEMBL7795914 0.91 TTR (0.43) TTRSLC6A2SLC6A3SLC6A4PTPRC
SCHEMBL7792631 0.89 HTR2A (0.39) TTRSLC6A2SLC6A3SLC6A4MEN1
SCHEMBL7796125 0.88 TTR (0.37) TTRSLC6A2SLC6A3SLC6A4PTPRC
SCHEMBL7794885 0.88 MEN1 (0.46) SLC6A2SLC6A3SLC6A4MEN1KMT2A
SCHEMBL7792655 0.86 HTR2A (0.40) TTRSLC6A2SLC6A3SLC6A4HTR2A
SCHEMBL7794729 0.86 TTR (0.38) TTRSLC6A2SLC6A3SLC6A4PTPRC
SCHEMBL7795927 0.86 TTR (0.38) TTRSLC6A2SLC6A3SLC6A4PTPRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906268-B1 ALKYLOXYAMINO SUBSTITUTED FLUORENONES AND THEIR USE AS PROTEIN KINASE C INHIBITORS AVENTIS PHARMA INC (US) 2001-11-28 EP disclosed
US-6004959-A HYPOTENSIVE, ANTITUMOR, ANTIINFLAMMATORY AND ANTIASTHMATIC AGENTS; ANGIOGENESIS AND ALVEOLAR MACROPHAGE ACTIVATION INHIBITORS HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US disclosed
EP-0906268-A1 ALKYLOXYAMINO SUBSTITUTED FLUORENONES AND THEIR USE AS PROTEIN KINASE C INHIBITORS HOECHST MARION ROUSSEL, INC. (US) 1999-04-07 EP disclosed
WO-1997045397-A1 ALKYLOXYAMINO SUBSTITUTED FLUORENONES AND THEIR USE AS PROTEIN KINASE C INHIBITORS HOECHST MARION ROUSSEL, INC. (US) 1997-12-04 WO disclosed