SCHEMBL7787003

SCHEMBL7787003

COc1cc2c(cc1Br)CC=C2CCNC(=O)C(F)(F)F

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 13/20 0.67
MTNR1B P49286 12/20 0.67
NQO2 P16083 9/20 0.67
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7784524 0.86 MTNR1A (0.50) MTNR1AMTNR1BNQO2
SCHEMBL7784807 0.84 MTNR1A (0.66) MTNR1AMTNR1BNQO2
SCHEMBL7785010 0.81 MTNR1A (1.00) MTNR1AMTNR1BNQO2
SCHEMBL25244513 0.77 HTR2A (0.58) MTNR1AMTNR1B
SCHEMBL7779907 0.74 NQO2 (0.65) MTNR1AMTNR1BNQO2
SCHEMBL16416372 0.73 CA12 (0.51)
Hydrochloric Acid SCHEMBL7784704 0.72 HTR2A (0.50) KDM4E
SCHEMBL7788014 0.72 NQO2 (0.54) MTNR1AMTNR1BNQO2
Hydrochloric Acid SCHEMBL7788560 0.72 MEN1 (0.41) MTNR1AMTNR1BNQO2
SCHEMBL27229051 0.71 MTNR1A (0.45) MTNR1AMTNR1BNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848699-B1 BENZOCYCLOALKENE COMPOUNDS WITH MELATONINE RECEPTOR BINDING AFFINITY, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-10-24 EP disclosed
US-5922771-A MELATONIN RECEPTOR AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-07-13 US disclosed
EP-0848699-A1 BENZOCYCLOALKENE COMPOUNDS WITH MELATONINE RECEPTOR BINDING AFFINITY, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-06-24 EP disclosed
WO-1997005098-A1 BENZOCYCLOALKENE COMPOUNDS WITH MELATONINE RECEPTOR BINDING AFFINITY, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-02-13 WO disclosed