SCHEMBL7787007

SCHEMBL7787007

COc1ccc2c(c1)N(C)c1ccccc1C2C(=O)Oc1c(F)cccc1F

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
MAPT P10636 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
TSHR P16473 4/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
CCKAR P32238 2/20 0.36
CCKBR P32239 2/20 0.36
RAB9A P51151 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 3/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
BCHE P06276 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL914119 0.92 HDAC4 (0.39) MEN1KMT2AMAPTHDAC4HDAC7
SCHEMBL5448645 0.89 HDAC4 (0.50) MEN1KMT2AMAPTHDAC4HDAC7
SCHEMBL38663637 0.89 HDAC4 (0.50) MEN1KMT2AMAPTHDAC4HDAC7
SCHEMBL7591680 0.86 SLC6A2 (0.37) MEN1KMT2AMAPTMAPK1RAB9A
SCHEMBL7031997 0.86 HDAC4 (0.45) MAPTHDAC4HDAC7HDAC5KDM4E
SCHEMBL7787045 0.86 HDAC4 (0.39) MEN1KMT2AMAPTHDAC4HDAC7
SCHEMBL14564649 0.83 MAPT (0.49) MEN1KMT2AMAPTHDAC4HDAC7
SCHEMBL38663301 0.82 HDAC4 (0.41) MEN1KMT2AMAPTHDAC4HDAC7
SCHEMBL8331335 0.82 MAPT (0.41) MAPTHDAC4HDAC7HDAC5KDM4E
SCHEMBL7592395 0.81 TAS1R3 (0.34) MEN1KMT2AMAPTLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0750748-B1 NOVEL ARYL N-ALKYLACRIDANCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN INC (US) 2001-12-05 EP claimed
EP-0750748-A4 NOVEL ARYL N-ALKYLACRIDANCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN INC (US) 1997-04-16 EP claimed
EP-0750748-A1 NOVEL ARYL N-ALKYLACRIDANCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN, INC. (US) 1997-01-02 EP claimed
WO-1995023971-A1 NOVEL ARYL N-ALKYLACRIDANCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN, INC. (US) 1995-09-08 WO claimed
US-20070059841-A1 ELECTROCHEMILUMINESCENCE FROM ACRIDAN COMPOUNDS LUMIGEN, INC. 2007-03-15 US disclosed
US-20070059841-A1 ELECTROCHEMILUMINESCENCE FROM ACRIDAN COMPOUNDS LUMIGEN, INC. 2007-03-15 US disclosed
US-7186568-B1 Providing a solution of an acridan compound and a peroxide, electrochemically oxidizing the acridan compound at a electrode to form an oxidized intermediate compound wherein the oxidized intermediate compound reacts with the peroxide provided in the solution to produce the chemiluminescence LUMIGEN INC. (US) 2007-03-06 US disclosed
US-7186568-B1 Providing a solution of an acridan compound and a peroxide, electrochemically oxidizing the acridan compound at a electrode to form an oxidized intermediate compound wherein the oxidized intermediate compound reacts with the peroxide provided in the solution to produce the chemiluminescence LUMIGEN INC. (US) 2007-03-06 US disclosed
EP-0750748-B1 NOVEL ARYL N-ALKYLACRIDANCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN INC (US) 2001-12-05 EP disclosed
US-5750698-A USEFUL IN DETECTING BOTH PEROXIDASE AND PEROXIDE LUMIGEN, INC. (US) 1998-05-12 US disclosed
EP-0750748-A4 NOVEL ARYL N-ALKYLACRIDANCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN INC (US) 1997-04-16 EP disclosed
US-5593845-A BY REACTION WITH PEROXIDES AND PEROXIDASE; DETECTION OF HAPTENS, PROTEINS, ANTIBODIES IN ENZYME IMMUNOASSAY LUMIGEN, INC. (US) 1997-01-14 US disclosed
EP-0750748-A1 NOVEL ARYL N-ALKYLACRIDANCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN, INC. (US) 1997-01-02 EP disclosed
WO-1995023971-A1 NOVEL ARYL N-ALKYLACRIDANCARBOXYLATE DERIVATIVES USEFUL FOR CHEMILUMINESCENT DETECTION LUMIGEN, INC. (US) 1995-09-08 WO disclosed