SCHEMBL7790201

SCHEMBL7790201

CCC#CC[C@@H]1C[C@@H](C(=O)OCc2ccccc2)N(C(=O)OC(C)(C)C)C1=O

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 5/20 0.40
KLK7 P49862 3/20 0.39
CTSL P07711 1/20 0.37
F2 P00734 2/20 0.37
KLK5 Q9Y337 2/20 0.37
CASP1 P29466 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7790190 0.93 KLK7 (0.40) FKBP1AKLK7CTSLF2KLK5
SCHEMBL7790063 0.91 FKBP1A (0.41) FKBP1AKLK7CTSLF2CASP1
SCHEMBL31486301 0.88 FKBP1A (0.44) FKBP1AKLK7CTSLF2KLK5
SCHEMBL22446555 0.86 KLK7 (0.45) FKBP1AKLK7CTSLF2KLK5
SCHEMBL30387086 0.86 KLK7 (0.45) FKBP1AKLK7CTSLF2KLK5
SCHEMBL31486524 0.86 KLK7 (0.45) FKBP1AKLK7CTSLF2KLK5
SCHEMBL12643706 0.86 KLK7 (0.45) FKBP1AKLK7CTSLF2KLK5
SCHEMBL23121510 0.84 FKBP1A (0.42) FKBP1AKLK7CTSLF2KLK5
SCHEMBL31486416 0.81 FKBP1A (0.45) FKBP1AKLK7CTSLF2HPGD
SCHEMBL31107722 0.81 FKBP1A (0.45) FKBP1AKLK7CTSLF2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0826663-B1 Alkynylamino acid derivatives and their use as pharmaceutical compounds LILLY CO ELI (GB) 2001-10-31 EP disclosed
EP-0826663-A2 Alkynylamino acid derivatives and their use as pharmaceutical compounds ELI LILLY AND COMPANY LIMITED (GB) 1998-03-04 EP disclosed