SCHEMBL7790532

SCHEMBL7790532

COc1cccc(CCNc2ccc(Cl)cc2)c1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.67
CHRM2 P08172 1/20 0.60
CHRM1 P11229 1/20 0.60
CHRM3 P20309 1/20 0.60
MAPT P10636 3/20 0.58
MEN1 O00255 1/20 0.58
KMT2A Q03164 1/20 0.58
HTT P42858 2/20 0.53
TAAR1 Q96RJ0 1/20 0.51
ACLY P53396 1/20 0.49
LMNA P02545 1/20 0.49
GAA P10253 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
DRD2 P14416 1/20 0.48
DRD4 P21917 1/20 0.48
BCHE P06276 1/20 0.48
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5517703 0.89 CHRM2 (0.66) CNR1CHRM2CHRM1CHRM3MAPT
SCHEMBL26268316 0.87 CHRM2 (0.67) CNR1CHRM2CHRM1CHRM3MAPT
SCHEMBL5115866 0.87 CHRM2 (0.62) CNR1CHRM2CHRM1CHRM3MAPT
SCHEMBL5101834 0.86 CHRM2 (0.66) CHRM2CHRM1CHRM3MEN1KMT2A
SCHEMBL19062086 0.85 CHRM2 (0.60) CNR1CHRM2CHRM1CHRM3MAPT
SCHEMBL5524054 0.84 CHRM2 (0.68) CNR1CHRM2CHRM1CHRM3MAPT
SCHEMBL30672995 0.84 CNR1 (0.58) CNR1CHRM2CHRM1CHRM3MAPT
SCHEMBL27904935 0.83 CHRM2 (0.66) CNR1CHRM2CHRM1CHRM3MEN1
SCHEMBL5108257 0.82 MEN1 (0.58) MAPTMEN1KMT2AHTTLMNA
SCHEMBL27922884 0.81 CHRM2 (0.59) CNR1CHRM2CHRM1CHRM3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021213358-A1 BORON-CONTAINING COMPOUNDS AND APPLICATION THEREOF 江苏先声药业有限公司 (CN) 2021-10-28 WO disclosed
EP-1150963-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM Aventis Pharma Deutschland GmbH (DE) 2001-11-07 EP disclosed
WO-2000046214-A1 SUBSTITUTED 4-AMINO-2-ARYLTETRAHYDROQUINAZOLINES, THEIR PREPARATION, THEIR USE AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-08-10 WO disclosed
US-4717724-A FUNGICIDES, ANTIPROTOZOA, BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1988-01-05 US disclosed
EP-0121753-A2 1-(1,3-Dioxolan-2-ylmethyl)-azoles, their salts, processes for their preparation and pharmaceutical compositions containing them HOECHST AKTIENGESELLSCHAFT (DE) 1984-10-17 EP disclosed