SCHEMBL7790590

SCHEMBL7790590

CCCC=Cc1cccc(F)c1F

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.40
TLR8 Q9NR97 1/20 0.40
NFE2L2 Q16236 10/20 0.39
ERN1 O75460 1/20 0.32
CHEK1 O14757 1/20 0.32
CDK4 P11802 1/20 0.32
CCNA2 P20248 1/20 0.32
CCND1 P24385 1/20 0.32
CDK2 P24941 1/20 0.32
CCND3 P30281 1/20 0.32
TRPA1 O75762 1/20 0.32
RELA Q04206 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7790587 1.00 PTGS2 (0.40) PTGS2TLR8NFE2L2ERN1CHEK1
SCHEMBL9419333 0.89 PDE5A (0.38) PTGS2NFE2L2
SCHEMBL9419329 0.89 PDE5A (0.38) PTGS2NFE2L2
SCHEMBL7530891 0.88 CYSLTR2 (0.40) PTGS2NFE2L2
SCHEMBL7530897 0.88 CYSLTR2 (0.40) PTGS2NFE2L2
SCHEMBL9419313 0.86 CYSLTR2 (0.42) PTGS2
SCHEMBL9419318 0.86 CYSLTR2 (0.42) PTGS2
SCHEMBL9419293 0.85 PTGS2 (0.42) PTGS2NFE2L2ERN1CHEK1CDK4
SCHEMBL9723201 0.85 PTGS2 (0.42) PTGS2NFE2L2ERN1CHEK1CDK4
SCHEMBL20640946 0.81 PTGS2 (0.40) PTGS2NFE2L2ERN1CHEK1CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144546-A3 FLUORINATED TERPHENYLS QinetiQ Limited (GB) 2002-08-28 EP disclosed
EP-1144546-A2 FLUORINATED TERPHENYLS QinetiQ Limited (GB) 2001-10-17 EP disclosed
WO-2000004111-A2 FLUORINATED TERPHENYLS THE SECRETARY OF STATE FOR DEFENCE (GB) 2000-01-27 WO disclosed
EP-0363458-B1 2,3-DIFLUOROBENZENES MERCK PATENT GMBH (DE) 1994-08-03 EP disclosed
US-5087764-A Deprotonation of a 1-substituted-2,3-difluorobenzene using an organometallic compound and reacting the reaction product with an electrophile Merck Patent Gesellschaft mit beschrankter Hafung (DE) 1992-02-11 US disclosed