Geclosporin

Geclosporin

SCHEMBL7791

C/C=C/CC(C)C(O)C1C(=O)NC(CCC)C(=O)N(C)CC(=O)N(C)C(CC(C)C)C(=O)NC(C(C)C)C(=O)N(C)C(CC(C)C)C(=O)NC(C)C(=O)NC(C)C(=O)N(C)C(CC(C)C)C(=O)N(C)C(CC(C)C)C(=O)N(C)C(C(C)C)C(=O)N1C

nearest known ligand 0.91

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 13/20 0.91
PPIA P62937 5/20 0.90
FKBP1B P68106 2/20 0.90
PPP3CA Q08209 2/20 0.90
MEN1 O00255 1/20 0.90
NPC1 O15118 1/20 0.90
ABCC3 O15438 1/20 0.90
GMNN O75496 1/20 0.90
USP2 O75604 1/20 0.90
SLCO2B1 O94956 1/20 0.90
ABCB11 O95342 1/20 0.90
LMNA P02545 1/20 0.90
POLB P06746 1/20 0.90
CYP3A4 P08684 1/20 0.90
MAPT P10636 1/20 0.90
RARB P10826 1/20 0.90
CYP2C9 P11712 1/20 0.90
CYP3A5 P20815 1/20 0.90
TACR2 P21452 1/20 0.90
PPIB P23284 1/20 0.90

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Geclosporin SCHEMBL2110698 1.00 ABCB1 (0.91) ABCB1PPIAFKBP1BPPP3CAMEN1
SCHEMBL18737282 0.96 ABCB1 (0.85) ABCB1PPIAFKBP1BPPP3CAMEN1
SCHEMBL23110295 0.96 PPIA (0.89) ABCB1PPIAFKBP1BPPP3CAMEN1
SCHEMBL16274167 0.95 ABCB1 (0.94) ABCB1PPIAFKBP1BPPP3CAMEN1
SCHEMBL17921935 0.95 ABCB1 (0.94) ABCB1PPIAFKBP1BPPP3CAMEN1
SCHEMBL13652544 0.95 ABCB1 (0.94) ABCB1PPIAFKBP1BPPP3CAMEN1
SCHEMBL22840735 0.95 ABCB1 (0.94) ABCB1PPIAFKBP1BPPP3CAMEN1
SCHEMBL23110210 0.95 ABCB1 (1.00) ABCB1PPIAFKBP1BPPP3CAMEN1
Cyclosporine SCHEMBL24239446 0.95 ABCB1 (1.00) ABCB1PPIAFKBP1BPPP3CAMEN1
Cyclosporine SCHEMBL24224445 0.95 ABCB1 (1.00) ABCB1PPIAFKBP1BPPP3CAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1817 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3641798-B1 COMPOSITIONS FOR THE PREVENTION AND TREATMENT OF ACUTE RENAL INJURY AKI THERAPEUTICS APS (DK) 2026-01-21 EP claimed
EP-3556774-B1 ANTI-CD40 ANTIBODIES AND USES THEREOF BETH ISRAEL DEACONESS MEDICAL CT INC (US) 2024-01-03 EP claimed
CN-116063481-A Humanized anti-CD 40 antibodies and uses thereof 普里玛托普医疗股份有限公司 2023-05-05 CN claimed
US-11471445-B2 Compositions for the prevention and treatment of acute renal injury AKI THERAPEUTICS APS (DK) 2022-10-18 US claimed
CN-109069621-B Humanized anti-CD 40 antibodies and uses thereof 普里玛托普医疗股份有限公司 2022-09-06 CN claimed
CN-114514019-A Method for producing pharmaceutical preparations containing crystalline and amorphous fractions of active substances 拜耳股份有限公司 2022-05-17 CN claimed
US-20210330649-A1 COMPOSITIONS FOR THE PREVENTION AND TREATMENT OF ACUTE RENAL INJURY AKI THERAPEUTICS APS (DK) 2021-10-28 US claimed
CN-112120033-A Application of ophiosporin G in preparation of marine fouling organism control agent 中国科学院南海海洋研究所 2020-12-25 CN claimed
EP-3641798-A1 COMPOSITIONS FOR THE PREVENTION AND TREATMENT OF ACUTE RENAL INJURY AKI THERAPEUTICS APS (DK) 2020-04-29 EP claimed
CN-110996985-A Composition for preventing and treating acute kidney injury AKI医疗有限公司 2020-04-10 CN claimed
EP-0512109-A1 ORAL PHARMACEUTICAL COMPOSITION CONTAINING CYCLOSPORIN AND PROCESS FOR PREPARING SAME. BIOGAL GYOGYSZERGYAR (HU) 1992-11-11 EP claimed
WO-1992018105-A1 IMPROVEMENTS IN PHARMACEUTICAL COMPOSITIONS SANDOZ LTD. (CH) 1992-10-29 WO claimed
EP-0506840-A1 METHOD OF TREATING OCULAR DISEASES BY PERIOCULAR ADMINISTRATION OF CYCLOSPORINE A OR G THE UNITED STATES OF AMERICA as represented by the Secretary United States Department of Commerce (US) 1992-10-07 EP claimed
WO-1992016226-A1 IL-1 INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1992-10-01 WO claimed
WO-1992009299-A1 ORAL PHARMACEUTICAL COMPOSITION CONTAINING CYCLOSPORIN AND PROCESS FOR PREPARING SAME BIOGAL Gyógyszergyár Rt. (HU) 1992-06-11 WO claimed
US-5051402-A Fungicides, immunosuppressants and antiphlogistic agents SANKYO COMPANY, LIMITED (JP) 1991-09-24 US claimed
US-5047396-A Cyclosporins, monester of hydroxylated fatty acid with ethylene glycol and mono or polyvalent alcohols BIOGAL GYOGYSZERGYAR (HU) 1991-09-10 US claimed
WO-1991008757-A1 METHOD OF TREATING OCULAR DISEASES BY PERIOCULAR ADMINISTRATION OF CYCLOSPORINE A OR G THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, U.S. DEPARTMENT OF COMMERCE (US) 1991-06-27 WO claimed
WO-1990000389-A1 FREEZE-DRIED LIPOSOME COMPOSITIONS CONTAINING CYCLOSPORIN REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 1990-01-25 WO claimed
US-4288431-A CULTURING TOLYPLOCLADIUM, CATALYTIC HYDROGENATION, REARRANGEMENT; ANTIINFLAMMATORY, IMMUNOLOGY SANDOZ LTD. (CH) 1981-09-08 US claimed