SCHEMBL7791758

SCHEMBL7791758

CCCC(=O)N[C@@H]1CCc2cc(OC)ccc2N(Cc2ccc(-c3ccccc3CNC(=O)NC)cc2)C1=O

nearest known ligand 0.63

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 4/20 0.63
XIAP P98170 10/20 0.48
AGTR1 P30556 1/20 0.42
NPY1R P25929 2/20 0.42
MTNR1A P48039 1/20 0.42
CCKBR P32239 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7795395 0.94 GHSR (0.65) GHSRXIAPAGTR1NPY1RMTNR1A
SCHEMBL7795638 0.94 GHSR (0.65) GHSRXIAPAGTR1NPY1RMTNR1A
SCHEMBL7786102 0.93 GHSR (0.64) GHSRXIAPAGTR1NPY1RMTNR1A
SCHEMBL7791537 0.92 GHSR (0.56) GHSRXIAPAGTR1NPY1RMTNR1A
SCHEMBL7791744 0.90 GHSR (0.65) GHSRXIAPAGTR1NPY1R
SCHEMBL7791562 0.90 GHSR (0.78) GHSRXIAPAGTR1NPY1R
SCHEMBL7796120 0.90 GHSR (0.69) GHSRXIAPAGTR1NPY1RMTNR1A
SCHEMBL7786051 0.89 GHSR (0.63) GHSRXIAPAGTR1NPY1R
SCHEMBL7795650 0.89 GHSR (0.81) GHSRXIAPAGTR1NPY1RCCKBR
SCHEMBL7791582 0.89 GHSR (0.66) GHSRXIAPAGTR1NPY1RMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0659179-B1 BENZO-FUSED LACTAMS PROMOTE RELEASE OF GROWTH HORMONE MERCK & CO INC (US) 2001-11-21 EP claimed
EP-0659179-B1 BENZO-FUSED LACTAMS PROMOTE RELEASE OF GROWTH HORMONE MERCK & CO INC (US) 2001-11-21 EP disclosed