SCHEMBL7791903

SCHEMBL7791903

Cc1cc(C)cc(CC(=O)N2CCCC(CCN3CCN(CC(C)C(=O)N(C)C)CC3)(c3ccc(Cl)c(Cl)c3)C2)c1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.48
TACR2 P21452 5/20 0.47
TACR1 P25103 5/20 0.47
TACR3 P29371 3/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5200433 0.85 CCR5 (0.51) CCR5TACR2TACR1TACR3CYP3A4
Hydrochloric Acid SCHEMBL6490695 0.84 CCR5 (0.50) CCR5TACR2TACR1TACR3CYP3A4
SCHEMBL5203138 0.82 TACR2 (0.51) CCR5TACR2TACR1TACR3CYP3A4
SCHEMBL5199990 0.81 CCR5 (0.54) CCR5TACR2TACR1TACR3CYP3A4
SCHEMBL5200438 0.80 SLC6A2 (0.51) CCR5TACR2TACR1TACR3CYP3A4
SCHEMBL5200182 0.80 TACR2 (0.52) CCR5TACR2TACR1TACR3
SCHEMBL5203186 0.79 CCR5 (0.54) CCR5TACR2TACR1TACR3
SCHEMBL5199904 0.78 CCR5 (0.53) CCR5TACR2TACR1TACR3CYP3A4
SCHEMBL5201070 0.78 CCR5 (0.49) CCR5TACR2TACR1TACR3CYP3A4
SCHEMBL5199623 0.78 CCR5 (0.53) CCR5TACR2TACR1TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150970-A1 (1-PHENACY-3-PHENYL-3-PIPERIDYLETHYL)PIPERIDINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME Sanofi-Aventis (FR) 2001-11-07 EP disclosed
WO-2000047572-A1 (1-PHENACY-3-PHENYL-3-PIPERIDYLETHYL)PIPERIDINE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SANOFI-SYNTHELABO (FR) 2000-08-17 WO disclosed