SCHEMBL7792601

SCHEMBL7792601

CCCOc1cc(OCC)c2c(c1)C(=O)c1cccc(OCCN3CCOCC3)c1-2

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 1/20 0.47
HTT P42858 1/20 0.47
MAPK14 Q16539 2/20 0.43
BRD4 O60885 1/20 0.43
NPC1 O15118 1/20 0.43
ADORA3 P0DMS8 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA2B P29275 1/20 0.42
ADORA1 P30542 1/20 0.42
TP53 P04637 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7792180 0.97 KDM4E (0.48) KDM4EALDH1A1HTTMAPK14BRD4
SCHEMBL7792176 0.97 KDM4E (0.50) KDM4EALDH1A1HTTMAPK14BRD4
SCHEMBL7786153 0.97 KDM4E (0.47) KDM4EALDH1A1HTTMAPK14BRD4
SCHEMBL7796357 0.97 KDM4E (0.47) KDM4EALDH1A1HTTMAPK14BRD4
SCHEMBL27495974 0.95 KDM4E (0.45) KDM4EALDH1A1HTTBRD4ADORA3
SCHEMBL7792104 0.95 KDM4E (0.50) KDM4EALDH1A1HTTMAPK14BRD4
SCHEMBL7786514 0.93 TSHR (0.46) KDM4EALDH1A1MAPK14TSHR
Hydrochloric Acid SCHEMBL7792093 0.92 ALDH1A1 (0.45) KDM4EALDH1A1TSHR
SCHEMBL7796433 0.92 ALDH1A1 (0.55) KDM4EALDH1A1HTTTSHR
SCHEMBL7796393 0.92 ALDH1A1 (0.52) KDM4EALDH1A1HTTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906268-B1 ALKYLOXYAMINO SUBSTITUTED FLUORENONES AND THEIR USE AS PROTEIN KINASE C INHIBITORS AVENTIS PHARMA INC (US) 2001-11-28 EP disclosed
US-6004959-A HYPOTENSIVE, ANTITUMOR, ANTIINFLAMMATORY AND ANTIASTHMATIC AGENTS; ANGIOGENESIS AND ALVEOLAR MACROPHAGE ACTIVATION INHIBITORS HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US disclosed