SCHEMBL7796341

SCHEMBL7796341

CCCOc1ccc2c(c1)C(=O)c1cccc(OCCN3CCOCC3)c1-2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.50
ADORA2A P29274 2/20 0.49
ADORA1 P30542 2/20 0.49
ADORA3 P0DMS8 1/20 0.49
ADORA2B P29275 1/20 0.49
NPC1 O15118 1/20 0.48
KDM4E B2RXH2 3/20 0.46
ALDH1A1 P00352 3/20 0.46
HTT P42858 1/20 0.46
PPARG P37231 1/20 0.46
CYP1A2 P05177 1/20 0.46
CHRM2 P08172 1/20 0.46
CHRM1 P11229 1/20 0.46
HTR2A P28223 1/20 0.46
MAPK1 P28482 1/20 0.46
SCN1A P35498 1/20 0.46
HTR2B P41595 1/20 0.46
KCNH2 Q12809 1/20 0.46
SCN2A Q99250 1/20 0.46
SIGMAR1 Q99720 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7786125 0.96 MAPK1 (0.51) MAPK14ADORA2AADORA1ADORA3ADORA2B
SCHEMBL7792021 0.93 KDM4E (0.52) MAPK14ADORA2AADORA1ADORA3ADORA2B
SCHEMBL7791807 0.92 ALDH1A1 (0.57) MAPK14KDM4EALDH1A1HTTCYP1A2
SCHEMBL7792420 0.91 HRH3 (0.51) ADORA2AADORA1KDM4EALDH1A1HRH3
SCHEMBL7786488 0.91 ADORA2A (0.56) MAPK14ADORA2AADORA1ADORA3ADORA2B
SCHEMBL7796357 0.90 KDM4E (0.47) MAPK14ADORA2AADORA1ADORA3ADORA2B
SCHEMBL7796315 0.90 CHEK1 (0.54) MAPK14ADORA2AADORA1ADORA3ADORA2B
SCHEMBL7786153 0.90 KDM4E (0.47) MAPK14ADORA2AADORA1ADORA3ADORA2B
SCHEMBL7786022 0.90 HRH3 (0.53) ADORA2AADORA1KDM4EALDH1A1HRH3
SCHEMBL7786514 0.88 TSHR (0.46) MAPK14KDM4EALDH1A1HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906268-B1 ALKYLOXYAMINO SUBSTITUTED FLUORENONES AND THEIR USE AS PROTEIN KINASE C INHIBITORS AVENTIS PHARMA INC (US) 2001-11-28 EP disclosed
US-6004959-A HYPOTENSIVE, ANTITUMOR, ANTIINFLAMMATORY AND ANTIASTHMATIC AGENTS; ANGIOGENESIS AND ALVEOLAR MACROPHAGE ACTIVATION INHIBITORS HOECHST MARION ROUSSEL, INC. (US) 1999-12-21 US disclosed