SCHEMBL7796763

SCHEMBL7796763

NC1=NC2(CCN(C(O)=S)CC2)Nc2cccc(F)c21

nearest known ligand 0.67

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 13/20 0.67
NOS1 P29475 11/20 0.67
NOS3 P29474 4/20 0.67
KCNH2 Q12809 1/20 0.41
DUSP3 P51452 1/20 0.32
PTPN5 P54829 1/20 0.32
PTPN11 Q06124 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HTR5A P47898 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
NEK2 P51955 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8376619 0.99 NOS2 (0.66) NOS2NOS1NOS3KCNH2DUSP3
Hydrochloric Acid SCHEMBL8378451 0.87 NOS2 (0.72) NOS2NOS1NOS3KCNH2HTR5A
SCHEMBL7796761 0.85 NOS2 (0.72) NOS2NOS1NOS3KCNH2HTR5A
SCHEMBL7931838 0.84 NOS2 (0.70) NOS2NOS1NOS3KCNH2ALDH1A1
Hydrochloric Acid SCHEMBL8379855 0.83 NOS2 (0.80) NOS2NOS1NOS3KCNH2KDM4E
Hydrochloric Acid SCHEMBL8380988 0.83 NOS2 (0.81) NOS2NOS1NOS3KCNH2KDM4E
Hydrochloric Acid SCHEMBL8376987 0.83 NOS2 (0.69) NOS2NOS1NOS3KCNH2ALDH1A1
SCHEMBL7803463 0.83 NOS2 (0.69) NOS2NOS1NOS3KCNH2NEK2
SCHEMBL8667931 0.83 NOS2 (0.65) NOS2NOS1NOS3KCNH2DUSP3
SCHEMBL7805035 0.82 NOS2 (0.81) NOS2NOS1NOS3KCNH2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248745-B1 MIXTURE COMPRISING A CYCLOOXYGENASE-2 (COX-2) INHIBITOR AND A 1,2-DIHYDRO-4-AMINOQUINAZOLINE DERIVATIVE INHIBITOR OF INDUCED NITRIC OXIDE SYNTHASE (INOS); NON-STEROIDAL ANTIINFLAMMATORY AGENTS ASTRAZENECA AB (SE) 2001-06-19 US claimed
EP-1100505-A1 A PHARMACEUTICAL COMBINATION COMPRISING A COX-2 INHIBITOR AND A iNOS INHIBITOR AstraZeneca AB (SE) 2001-05-23 EP claimed
WO-2000000200-A1 A PHARMACEUTICAL COMBINATION COMPRISING A COX-2 INHIBITOR AND A iNOS INHIBITOR ASTRAZENECA AB (SE) 2000-01-06 WO claimed