SCHEMBL7797012

SCHEMBL7797012

CC(C)(C)OC(=O)N=C(N)N(C(=O)OC(C)(C)C)c1cccc(C=O)c1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
UNG P13051 1/20 0.32
NR1H4 Q96RI1 4/20 0.32
BRD4 O60885 1/20 0.31
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
SLC9A1 P19634 1/20 0.31
SLC9A3 P48764 1/20 0.31
SLC9A2 Q9UBY0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3119357 0.85 UNG (0.40) UNGNR1H4BRD4NPC1MAPT
SCHEMBL3785117 0.82 KMT2A (0.34) BRD4MAPTRAB9ASMN1; SMN2
SCHEMBL15140038 0.82 F2 (0.35) BRD4NPC1RAB9A
SCHEMBL207903 0.81 MTNR1B (0.35) BRD4
SCHEMBL6701854 0.80 MAPT (0.43) NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL3688119 0.79 ITGB1 (0.31) BRD4
SCHEMBL3778075 0.78 TP53 (0.31) MAPT
SCHEMBL17894521 0.76 MIF (0.36)
SCHEMBL208845 0.76 HDAC3 (0.33)
SCHEMBL3777967 0.76 SCN2A (0.32) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159260-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-05 EP claimed
WO-2000055124-A2 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO claimed
EP-1159260-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000055124-A2 NOVEL COMPOUNDS AND COMPOSITIONS AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed