SCHEMBL7797261

SCHEMBL7797261

CCOC(=O)c1c(-c2ccncc2)c(-c2ccc(S(N)(=O)=O)cc2)nn1C

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 12/20 0.50
CA12 O43570 5/20 0.50
CHRNA7 P36544 3/20 0.46
CA1 P00915 5/20 0.46
CA2 P00918 5/20 0.46
CA4 P22748 4/20 0.45
PTGS1 P23219 1/20 0.45
PTGS2 P35354 1/20 0.45
MAPK13 O15264 1/20 0.43
MAPK12 P53778 1/20 0.43
MAPK11 Q15759 1/20 0.43
MAPK14 Q16539 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8168023 1.00 CA9 (0.50) CA9CA12CHRNA7CA1CA2
SCHEMBL8181215 0.90 CA12 (0.48) CA9CA12PTGS2MAPK13MAPK12
SCHEMBL8176091 0.90 CA12 (0.48) CA9CA12PTGS2MAPK13MAPK12
SCHEMBL8181108 0.88 CA12 (0.47) CA9CA12CA1CA2PTGS1
SCHEMBL7799176 0.88 CA12 (0.47) CA9CA12CA1CA2PTGS1
SCHEMBL8174257 0.87 ALDH1A1 (0.47) CA9CA12CA1CA2CA4
SCHEMBL8181992 0.87 ALDH1A1 (0.47) CA9CA12CA1CA2CA4
SCHEMBL8174276 0.85 TP53 (0.46) CA9CA12CA1CA2PTGS1
SCHEMBL8175722 0.85 TP53 (0.46) CA9CA12CA1CA2PTGS1
SCHEMBL7779780 0.84 IKBKB (0.46) CA9CA12CA1CA2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0772597-B1 3,4-SUBSTITUTED PYRAZOLES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2001-12-12 EP claimed
US-6028072-A 3,4-substituted pyrazoles for the treatment of inflammation G. D. SEARLE & CO. (US) 2000-02-22 US claimed