SCHEMBL7800224

SCHEMBL7800224

C#CC(Cc1ccccc1)NCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.53
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
TSHR P16473 1/20 0.49
MAOB P27338 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.42
LMNA P02545 1/20 0.40
IDO1 P14902 2/20 0.39
THRB P10828 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
EPHX1 P07099 1/20 0.39
POLB P06746 1/20 0.39
ACP3 P15309 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21153206 0.84 SLC1A1 (0.43) SIGMAR1MAOBLMNAIDO1POLB
SCHEMBL26858667 0.84 CYP2D6 (0.43) SIGMAR1CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL896529 0.83 SIGMAR1 (0.56) SIGMAR1CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL21153204 0.81 CASR (0.56) MAOBSMN1; SMN2IDO1MEN1KMT2A
SCHEMBL3177171 0.79 ACE (0.47) CYP1A2CYP3A4CYP2D6TSHRMEN1
SCHEMBL25208573 0.79 MEN1 (0.53) CYP3A4CYP2D6TSHRMEN1KMT2A
SCHEMBL1716115 0.74 SIGMAR1 (0.55) SIGMAR1CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL17865679 0.74 CTSC (0.50) CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL1519814 0.74 CTSC (0.50) CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL4901736 0.74 CTSC (0.50) CYP1A2CYP3A4CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0748801-B1 2-ISOXAZOLINE DERIVATIVE AND PROCESS FOR PRODUCING THE SAME, AND PROCESS FOR PRODUCING RELATED DERIVATIVES FROM THE SAME DAICEL CHEM (JP) 2001-12-19 EP disclosed
US-6018069-A 2-isoxazoline derivative and process for producing the same and process for producing related derivatives from the same DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 2000-01-25 US disclosed
US-5994558-A 2-isoxazoline derivative and process for producing the same; and process for producing related derivatives from the same DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1999-11-30 US disclosed
US-5962692-A 2-isoxazoline derivative and process for producing the same, and process for producing related derivatives from the same DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1999-10-05 US disclosed
US-5750717-A 2-isoxazoline derivative and process for producing the same, and process for producing related derivatives from the same DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-12 US disclosed
EP-0748801-A1 2-ISOXAZOLINE DERIVATIVE AND PROCESS FOR PRODUCING THE SAME, AND PROCESS FOR PRODUCING RELATED DERIVATIVES FROM THE SAME DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-18 EP disclosed