SCHEMBL7801877

SCHEMBL7801877

Cc1ccc(C(O)(COC(=O)C(C)C)COC(=O)C(C)C)c(C)c1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.76
MAPT P10636 3/20 0.76
POLB P06746 2/20 0.76
CYP2C9 P11712 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPSR1 Q6W5P4 1/20 0.38
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
LMNA P02545 2/20 0.36
GPR55 Q9Y2T6 1/20 0.36
KDM4E B2RXH2 2/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GAA P10253 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
TAS1R2 Q8TE23 1/20 0.33
HTT P42858 1/20 0.33
APEX1 P27695 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8528468 0.87 ALDH1A1 (1.00) ALDH1A1MAPTPOLBCYP2C9NPSR1
SCHEMBL7808592 0.81 ALDH1A1 (0.58) ALDH1A1MAPTPOLBSMN1; SMN2NPSR1
SCHEMBL26261032 0.80 ALDH1A1 (0.87) ALDH1A1MAPTPOLBCYP2C9SMN1; SMN2
SCHEMBL7808248 0.78 MAPT (0.61) ALDH1A1MAPTPOLBCYP2C9NPSR1
Acetic Acid SCHEMBL7949781 0.77 POLB (0.81) ALDH1A1MAPTPOLBCYP2C9SMN1; SMN2
SCHEMBL7949793 0.77 ALDH1A1 (0.81) ALDH1A1MAPTPOLBCYP2C9SMN1; SMN2
SCHEMBL7949777 0.76 POLB (0.60) ALDH1A1MAPTPOLBCYP2C9SMN1; SMN2
SCHEMBL7801666 0.75 ALDH1A1 (0.58) ALDH1A1MAPTPOLBCYP2C9NPSR1
SCHEMBL7811026 0.75 ALDH1A1 (0.58) ALDH1A1MAPTPOLBCYP2C9SMN1; SMN2
SCHEMBL8147616 0.72 MAPT (0.55) ALDH1A1MAPTPOLBCYP2C9SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1120397-A2 Process for preparing triazole derivative KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 2001-08-01 EP disclosed
EP-0704419-B1 PROCESS FOR PRODUCING AN OPTICALLY ACTIVE 2-ARYL-3-ACYLOXY-1,2-PROPANEDIOL KANEGAFUCHI CHEMICAL IND (JP) 2001-07-25 EP disclosed
US-6046354-A CHEMICAL INTERMEDIATES, E.G. 2-ARYL-1,3-DIACYLOXY-2-PROPANOL, FOR DRUGS AND FUNGICIDES,E.G. (R)-2-(2,4-DIFLUOROPHENYL)-3-(1H-1,2,4-TRIAZOLE-1-YL)-PROPANE-1,2-DIOL, KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 2000-04-04 US disclosed
US-5840553-A OPTICALLY ACTIVE 2-ARYL-3-ACYLOXY-1,2,-PROPANE DIOL USING A MICROORGANISM OR ENZYME DERIVED FROM PORCINE PANCREAS; VIA STEREOSPECIFIC HYDROLYSIS OF A 2-ARYL-1,3-DIACYLOXY-2-PROPANOL; SYNTHETIC CHEMICAL INTERMEDIATES, FUNGICIDES KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1998-11-24 US disclosed
US-5654472-A OPTICALLY PURE 2-ARYL-3-ACYLOXY-1,2-PROPANEDIOL COMPOUNDS; CHEMICAL INTERMEDIATES KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1997-08-05 US disclosed
EP-0704419-A1 PROCESS FOR PRODUCING TRIAZOLE DERIVATIVE KANEGAFUCHI KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1996-04-03 EP disclosed