SCHEMBL7801951

SCHEMBL7801951

C1=C(COCc2ccccc2)CCNC1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.50
SIGMAR1 Q99720 1/20 0.44
HTR2C P28335 3/20 0.43
TACR1 P25103 1/20 0.42
HTR2B P41595 1/20 0.38
HTR1A P08908 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
HTR2A P28223 1/20 0.38
PRMT5 O14744 3/20 0.37
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
QDPR P09417 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7404347 0.79 SIGMAR1 (0.50) TSHRSIGMAR1HTR2CHTR2BHTR1A
SCHEMBL28713802 0.78 TSHR (0.62) TSHRTACR1
SCHEMBL15004237 0.78 SIGMAR1 (0.46) SIGMAR1HTR2CHTR1ASLC6A2SLC6A4
Hydrochloric Acid SCHEMBL1574641 0.77 HTR2C (0.52) TSHRSIGMAR1HTR2CHTR2BHTR1A
Hydrochloric Acid SCHEMBL14995164 0.77 HTR2C (0.47) SIGMAR1HTR2CHTR1ASLC6A2SLC6A4
Hydrochloric Acid SCHEMBL14995271 0.76 HTR2C (0.50) SIGMAR1HTR2CHTR2B
SCHEMBL11633937 0.75 SIGMAR1 (0.46) SIGMAR1HTR2C
SCHEMBL11633520 0.75 SIGMAR1 (0.46) SIGMAR1HTR2CHTR2A
SCHEMBL18989466 0.74 TSHR (0.56) TSHRHTR1A
SCHEMBL9725547 0.73 TSHR (0.94) TSHRTACR1SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024039829-A1 INHIBITORS OF KIF18A AND USES THEREOF ACCENT THERAPEUTICS, INC. (US) 2024-02-22 WO disclosed
EP-0873317-B1 PYRIMIDIN DERIVATIVES HOFFMANN LA ROCHE (CH) 2001-04-11 EP disclosed
EP-0873317-A1 PYRIMIDIN DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1998-10-28 EP disclosed
US-5688798-A PSYCHOTIC ILLNESS SUCH AS SCHIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1997-11-18 US disclosed
WO-1997013759-A1 PYRIMIDIN DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-04-17 WO disclosed