SCHEMBL7802933

SCHEMBL7802933

NC1=NC2(CCCN(Cc3ccccc3)C2)Nc2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 7/20 0.47
NOS2 P35228 2/20 0.42
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CYP3A4 P08684 4/20 0.40
TSHR P16473 4/20 0.40
GAA P10253 2/20 0.40
POLB P06746 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HSD17B10 Q99714 1/20 0.39
SIGMAR1 Q99720 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8379804 0.99 CYP2D6 (0.46) CYP2D6NOS2ALDH1A1KDM4ELMNA
SCHEMBL7805049 0.93 POLB (0.44) CYP2D6NOS2ALDH1A1KDM4ELMNA
Hydrochloric Acid SCHEMBL8379825 0.92 POLB (0.43) CYP2D6NOS2ALDH1A1KDM4ELMNA
SCHEMBL7796674 0.85 POLB (0.49) NOS2ALDH1A1KDM4ELMNAHTT
Hydrochloric Acid SCHEMBL8380986 0.84 POLB (0.48) NOS2ALDH1A1KDM4ELMNAHTT
SCHEMBL7796701 0.77 NOS2 (0.57) NOS2ALDH1A1KDM4ELMNAHTT
SCHEMBL7796722 0.76 NOS2 (0.56) NOS2ALDH1A1KDM4ELMNAHTT
Hydrochloric Acid SCHEMBL8380958 0.76 NOS2 (0.56) NOS2ALDH1A1KDM4ELMNAHTT
Hydrochloric Acid SCHEMBL8377757 0.75 NOS2 (0.54) NOS2ALDH1A1KDM4ELMNAHTT
SCHEMBL7940895 0.73 NOS2 (0.55) NOS2ALDH1A1KDM4ELMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248745-B1 MIXTURE COMPRISING A CYCLOOXYGENASE-2 (COX-2) INHIBITOR AND A 1,2-DIHYDRO-4-AMINOQUINAZOLINE DERIVATIVE INHIBITOR OF INDUCED NITRIC OXIDE SYNTHASE (INOS); NON-STEROIDAL ANTIINFLAMMATORY AGENTS ASTRAZENECA AB (SE) 2001-06-19 US claimed
EP-1100505-A1 A PHARMACEUTICAL COMBINATION COMPRISING A COX-2 INHIBITOR AND A iNOS INHIBITOR AstraZeneca AB (SE) 2001-05-23 EP claimed
WO-2000000200-A1 A PHARMACEUTICAL COMBINATION COMPRISING A COX-2 INHIBITOR AND A iNOS INHIBITOR ASTRAZENECA AB (SE) 2000-01-06 WO claimed