SCHEMBL7803012

SCHEMBL7803012

COc1ccc(CN(C)C(=O)CC(CC=O)c2ccc(Cl)c(Cl)c2)cc1F

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.44
MITF O75030 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HTT P42858 1/20 0.44
CDK8 P49336 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
FFAR1 O14842 1/20 0.40
CXCR3 P49682 6/20 0.39
HSP90AA1 P07900 1/20 0.38
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7812269 0.89 FFAR1 (0.48) KDM4EMITFALDH1A1HTTCDK8
SCHEMBL7807544 0.88 KDM4E (0.45) KDM4EMITFALDH1A1HTTCDK8
SCHEMBL7815283 0.88 KDM4E (0.45) KDM4EMITFALDH1A1HTTCDK8
SCHEMBL7815281 0.84 FFAR1 (0.44) KDM4EMITFALDH1A1HTTCDK8
SCHEMBL7807790 0.83 TACR1 (0.55) ALDH1A1HTTCDK8CLK4HSP90AA1
SCHEMBL7809517 0.83 TACR1 (0.47) ALDH1A1TDP1
SCHEMBL6961996 0.82 MEN1 (0.47) TDP1
SCHEMBL7811343 0.81 TACR1 (0.49) HTTHSP90AA1TDP1
SCHEMBL7807768 0.80 TACR1 (0.44) ALDH1A1TDP1
SCHEMBL7803017 0.79 KDM4E (0.43) KDM4EMITFALDH1A1HTTCDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773929-B1 PIPERIDINE DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORP (US) 2001-10-31 EP disclosed
US-5654316-A Piperidine derivatives as neurokinin antagonists SCHERING CORPORATION (US) 1997-08-05 US disclosed