SCHEMBL7811343

SCHEMBL7811343

CN(Cc1ccccc1)C(=O)CC(CC=O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.49
LMNA P02545 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
HTT P42858 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
TDP1 Q9NUW8 1/20 0.43
HPGD P15428 1/20 0.43
SLC6A4 P31645 1/20 0.42
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42
HSP90AA1 P07900 1/20 0.41
TACR2 P21452 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7809427 0.87 TACR1 (0.52) TACR1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL7809517 0.87 TACR1 (0.47) TACR1LMNAKMT2AMEN1TDP1
SCHEMBL7815209 0.85 TACR1 (0.50) TACR1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL7807790 0.85 TACR1 (0.55) TACR1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL7807768 0.84 TACR1 (0.44) TACR1LMNAKMT2AMEN1TDP1
SCHEMBL7811404 0.84 TACR1 (0.49) TACR1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL6969734 0.84 ALDH1A1 (0.49) TACR1CYP3A4CYP2D6KMT2AMEN1
SCHEMBL6961996 0.83 MEN1 (0.47) TACR1CYP3A4CYP2D6KMT2AMEN1
SCHEMBL8801314 0.81 HPGD (0.45) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8801310 0.81 HPGD (0.45) LMNACYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773929-B1 PIPERIDINE DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORP (US) 2001-10-31 EP disclosed
US-5654316-A Piperidine derivatives as neurokinin antagonists SCHERING CORPORATION (US) 1997-08-05 US disclosed