SCHEMBL7804069

SCHEMBL7804069

F[B]F.Nc1c(F)c(F)c(OC(F)F)c2c1c(=O)c(C(=O)O)cn2C1CC1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 17/20 0.57
CACNA1F O60840 1/20 0.53
POLB P06746 1/20 0.53
MAPK1 P28482 1/20 0.53
CACNA1D Q01668 1/20 0.53
KCNH2 Q12809 1/20 0.53
CACNA1S Q13698 1/20 0.53
CACNA1C Q13936 1/20 0.53
TOP2A P11388 1/20 0.52
TOP2B Q02880 1/20 0.52
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1986275 0.97 GSK3B (0.60) GSK3BCACNA1FPOLBMAPK1CACNA1D
Fluoride SCHEMBL7804066 0.95 GSK3B (0.58) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL1343006 0.88 GSK3B (0.65) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL500863 0.84 GSK3B (0.64) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL7810902 0.83 GSK3B (0.48) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL9689537 0.82 GSK3B (0.68) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL7812725 0.82 CACNA1F (0.57) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL7816829 0.82 KCNH2 (0.57) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL7813328 0.81 KCNH2 (0.56) GSK3BCACNA1FPOLBMAPK1CACNA1D
SCHEMBL1345769 0.81 GSK3B (0.70) GSK3BCACNA1FPOLBMAPK1CACNA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0610958-B1 Intermediates in the preparation of 4-oxoquinoline-3-carboxylic acid derivatives UBE INDUSTRIES (JP) 2001-10-04 EP disclosed
US-5496951-A 1-CYCLOPROPYL-6-FLUORO-8-FLUORINATED METHOXY COMPOUNDS INCLUDING BORON DIFLUORIDE CHELATE; CHEMICAL INTERMEDIATES AND ANTIBACTERIAL AGENTS SANKYO COMPANY, LIMITED (JP) 1996-03-05 US disclosed
US-5436367-A 3, 4-difluorobenzoic acid derivatives SANKO COMPANY, LIMITED (JP) 1995-07-25 US disclosed
EP-0352123-B1 4-Oxoquinoline-3-carboxylic acid derivatives, their preparation and their use UBE INDUSTRIES (JP) 1995-01-18 EP disclosed
US-5348961-A Antibacterial agents SANKYO COMPANY LIMITED (JP) 1994-09-20 US disclosed
EP-0610958-A2 Intermediates in the preparation of 4-oxoquinoline-3-carboxylic acid derivatives UBE INDUSTRIES, LTD. (JP) 1994-08-17 EP disclosed
US-5073556-A Bactericides SANKYO COMPANY LIMITED (JP) 1991-12-17 US disclosed
EP-0352123-A2 4-Oxoquinoline-3-carboxylic acid derivatives, their preparation and their use UBE INDUSTRIES LIMITED (JP) 1990-01-24 EP disclosed