SCHEMBL7804282

SCHEMBL7804282

C[C@H](O)CCCCOc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA3 P22001 1/20 0.61
LMNA P02545 1/20 0.60
CHRNB2 P17787 2/20 0.52
CHRNB4 P30926 2/20 0.52
CHRNA3 P32297 2/20 0.52
CHRNA7 P36544 2/20 0.52
CHRNA4 P43681 2/20 0.52
LTA4H P09960 2/20 0.50
ALDH1A1 P00352 1/20 0.50
RECQL P46063 1/20 0.50
HDAC3 O15379 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC10 Q969S8 1/20 0.50
HDAC11 Q96DB2 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
HDAC9 Q9UKV0 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6247219 1.00 KCNA3 (0.61) KCNA3LMNACHRNB2CHRNB4CHRNA3
SCHEMBL17201876 0.98 KCNA3 (0.59) KCNA3LMNACHRNB2CHRNB4CHRNA3
SCHEMBL166338 0.88 LMNA (0.64) KCNA3LMNACHRNB2CHRNB4CHRNA3
SCHEMBL11580701 0.84 KCNA3 (0.67) KCNA3LMNALTA4HALDH1A1RECQL
SCHEMBL7804270 0.83 MEN1 (0.53) ALDH1A1MEN1KMT2AHPGDRARB
SCHEMBL8755014 0.83 HPGD (0.49) CHRNB4CHRNA3CHRNA7ALDH1A1TDP1
SCHEMBL12746095 0.82 KCNA3 (0.64) KCNA3LMNALTA4HHDAC3HDAC4
SCHEMBL358609 0.82 KCNA3 (0.64) KCNA3LMNALTA4HHDAC3HDAC4
SCHEMBL11068531 0.82 KCNA3 (0.64) KCNA3LMNALTA4HHDAC3HDAC4
SCHEMBL13829034 0.82 LMNA (0.62) LMNAALDH1A1RECQLMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1104395-A1 STEREOSELECTIVE RING OPENING REACTIONS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2001-06-06 EP disclosed
WO-2000009463-A1 STEREOSELECTIVE RING OPENING REACTIONS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2000-02-24 WO disclosed