SCHEMBL7804897

SCHEMBL7804897

C=C(Br)C(=O)Nc1cc(C(=O)Nc2cc(C(=O)Nc3c[nH]c(C(=O)NCCC#N)c3C)n(C)c2)n(C)c1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 2/20 0.38
HRAS P01112 2/20 0.38
ESR1 P03372 2/20 0.38
ESR2 Q92731 2/20 0.38
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
HIF1A Q16665 1/20 0.37
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC8 Q9BY41 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7800926 0.88 HRAS (0.40) TOP1HRASESR1ESR2KDM4E
SCHEMBL7118414 0.86 HRAS (0.48) TOP1HRASESR1ESR2KDM4E
SCHEMBL7117804 0.86 HRAS (0.48) TOP1HRASESR1ESR2KDM4E
SCHEMBL8444844 0.85 GRM1 (0.32)
SCHEMBL8442943 0.85 GRM1 (0.32)
SCHEMBL7647214 0.84 HRAS (0.45) TOP1HRASESR1ESR2KDM4E
SCHEMBL7803321 0.82 TOP1 (0.43) TOP1HRASESR1ESR2KDM4E
SCHEMBL7645811 0.80 TOP1 (0.37) TOP1HRASESR1ESR2KDM4E
SCHEMBL7813677 0.78 ITGB3 (0.35) KDM4EMAPTHDAC1
SCHEMBL6781964 0.78 HRAS (0.43) TOP1HRASESR1ESR2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915845-B1 ACRYLOYL SUBSTITUTED DISTAMYCIN DERIVATIVES, PROCESS FOR PREPARING THEM, AND THEIR USE AS ANTITUMOR AND ANTIVIRAL AGENTS PHARMACIA & UPJOHN SPA (IT) 2001-09-12 EP disclosed