SCHEMBL7806768

SCHEMBL7806768

CCOC(=O)NC(CC)C1N=C(N)c2ccccc2N1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 2/20 0.44
KDM4E B2RXH2 13/20 0.43
ALDH1A1 P00352 13/20 0.43
GAA P10253 6/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
HPGD P15428 4/20 0.41
THRB P10828 3/20 0.41
POLB P06746 1/20 0.39
KMT2A Q03164 1/20 0.38
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8377836 0.99 NOS2 (0.43) NOS2KDM4EALDH1A1GAASMN1; SMN2
Hydrochloric Acid SCHEMBL8379182 0.86 NOS2 (0.44) NOS2KDM4EALDH1A1GAASMN1; SMN2
SCHEMBL7806671 0.75 NOS2 (0.57) NOS2KDM4EALDH1A1GAASMN1; SMN2
SCHEMBL7806698 0.74 NOS2 (0.54) NOS2KDM4EALDH1A1GAASMN1; SMN2
Hydrochloric Acid SCHEMBL8379186 0.73 NOS2 (0.53) NOS2KDM4EALDH1A1GAASMN1; SMN2
SCHEMBL7806770 0.72 NOS2 (0.52) NOS2KDM4EALDH1A1GAASMN1; SMN2
Hydrochloric Acid SCHEMBL8377837 0.71 NOS2 (0.51) NOS2KDM4EALDH1A1GAASMN1; SMN2
SCHEMBL7938417 0.66 NOS2 (0.45) NOS2KDM4EALDH1A1GAASMN1; SMN2
Hydrochloric Acid SCHEMBL8376464 0.65 NOS2 (0.44) NOS2KDM4EALDH1A1GAASMN1; SMN2
Hydrochloric Acid SCHEMBL8382185 0.62 NOS2 (0.97) NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248745-B1 MIXTURE COMPRISING A CYCLOOXYGENASE-2 (COX-2) INHIBITOR AND A 1,2-DIHYDRO-4-AMINOQUINAZOLINE DERIVATIVE INHIBITOR OF INDUCED NITRIC OXIDE SYNTHASE (INOS); NON-STEROIDAL ANTIINFLAMMATORY AGENTS ASTRAZENECA AB (SE) 2001-06-19 US claimed
EP-1100505-A1 A PHARMACEUTICAL COMBINATION COMPRISING A COX-2 INHIBITOR AND A iNOS INHIBITOR AstraZeneca AB (SE) 2001-05-23 EP claimed
WO-2000000200-A1 A PHARMACEUTICAL COMBINATION COMPRISING A COX-2 INHIBITOR AND A iNOS INHIBITOR ASTRAZENECA AB (SE) 2000-01-06 WO claimed