SCHEMBL7808154

SCHEMBL7808154

CN1C(=O)C(NC(=O)C(N)Cc2ccccc2)N=C(N2CC3CCC(CC3)C2)c2ccccc21

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 11/20 0.68
KCNH2 Q12809 1/20 0.68
SCN9A Q15858 5/20 0.50
CCKAR P32238 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9526270 0.81 CCKBR (1.00) CCKBRKCNH2SCN9ACCKAR
SCHEMBL9526276 0.81 CCKBR (1.00) CCKBRKCNH2SCN9ACCKAR
SCHEMBL9525366 0.81 CCKBR (1.00) CCKBRKCNH2SCN9ACCKAR
SCHEMBL9525360 0.81 CCKBR (1.00) CCKBRKCNH2SCN9ACCKAR
SCHEMBL8880870 0.81 CCKBR (0.69) CCKBRKCNH2SCN9A
SCHEMBL8880864 0.81 CCKBR (0.69) CCKBRKCNH2SCN9A
SCHEMBL9008767 0.81 CCKBR (0.69) CCKBRKCNH2SCN9A
SCHEMBL9008763 0.81 CCKBR (0.69) CCKBRKCNH2SCN9A
SCHEMBL8879465 0.81 CCKBR (0.69) CCKBRKCNH2SCN9A
SCHEMBL9303610 0.81 CCKBR (0.69) CCKBRKCNH2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0652871-B1 BENZODIAZEPINE DERIVATIVES MERCK SHARP & DOHME (GB) 2001-10-17 EP disclosed
US-5618812-A GASTRIN ANTAGONISTS; GASTROINTESTINAL DISORDERS MERCK SHARP & DOHME, LTD. (GB) 1997-04-08 US disclosed