SCHEMBL7808378

SCHEMBL7808378

Cc1cc(N(C(=O)CCNC(=O)OC(C)(C)C)C(C)C)c(C)cc1C#CCNc1ccc(C(=N)N)cc1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
PTPN11 Q06124 1/20 0.33
F2 P00734 4/20 0.32
TMPRSS6 Q8IU80 4/20 0.32
PRMT1 Q99873 1/20 0.31
ITGB3 P05106 4/20 0.30
ITGA2B P08514 4/20 0.30
MALT1 Q9UDY8 1/20 0.30
PLAU P00749 1/20 0.30
ATR Q13535 1/20 0.30
AAK1 Q2M2I8 1/20 0.30
HPN P05981 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6562003 0.92 PTPN11 (0.33) CA1CA2PTPN11MALT1AAK1
SCHEMBL6565916 0.85 ITGB3 (0.35) F2ITGB3ITGA2BPLAUHPN
SCHEMBL6562499 0.85 ITGB3 (0.34) F2TMPRSS6ITGB3ITGA2BPLAU
SCHEMBL6563611 0.84 ITGB3 (0.38) F2ITGB3ITGA2BPLAU
SCHEMBL6561908 0.84 PTPN11 (0.33) PTPN11AAK1
SCHEMBL6563607 0.84 ITGB3 (0.40) F2ITGB3ITGA2BPLAU
SCHEMBL6561947 0.83 F10 (0.36) F2ITGB3ITGA2BPLAU
SCHEMBL6561873 0.83 ITGB3 (0.38) F2ITGB3ITGA2B
SCHEMBL4250003 0.82 ITGB3 (0.37) F2TMPRSS6ITGB3ITGA2BPLAU
SCHEMBL6563542 0.82 ITGB3 (0.37) F2ITGB3ITGA2BPLAUHPN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM KG (DE) 2001-10-10 EP disclosed
WO-2000035859-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-06-22 WO disclosed