SCHEMBL7808388

SCHEMBL7808388

CCCCOC(=O)N=C(N)c1ccc(NCC#Cc2ccc(C(=O)N3CCCC3C(OC)C(=O)OCC)c(C)c2)cc1

nearest known ligand 0.32

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.32
F2 P00734 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
SLC6A2 P23975 1/20 0.32
AGTR1 P30556 1/20 0.32
SLC6A3 Q01959 1/20 0.32
SCN5A Q14524 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
GAA P10253 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ITGB3 P05106 2/20 0.30
ITGA2B P08514 2/20 0.30
ALDH1A1 P00352 2/20 0.30
ADRB2 P07550 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7806152 0.88 HRH3 (0.37) NR1I2F2ADORA3SLC6A2AGTR1
SCHEMBL6565376 0.86 PRSS1 (0.35) F2GAASMN1; SMN2ITGB3ITGA2B
SCHEMBL7806160 0.86 MEN1 (0.40) NR1I2F2ADORA3SLC6A2AGTR1
SCHEMBL7809950 0.82 PIK3CA (0.40) NR1I2F2ADORA3SLC6A2AGTR1
SCHEMBL7804851 0.81 HRH3 (0.36) L3MBTL1
SCHEMBL7809959 0.80 SMN1; SMN2 (0.39) NR1I2F2ADORA3SLC6A2AGTR1
SCHEMBL7804870 0.79 HRH3 (0.43) L3MBTL1GAAALDH1A1HPGD
SCHEMBL6563725 0.79 GAA (0.33) GAASMN1; SMN2ALDH1A1
SCHEMBL6565851 0.79 F2 (0.37) F2GAASMN1; SMN2ITGB3ITGA2B
SCHEMBL7806863 0.78 HRH3 (0.35) NR1I2F2ADORA3SLC6A2AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM KG (DE) 2001-10-10 EP disclosed
WO-2000035859-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-06-22 WO disclosed