SCHEMBL6563725

SCHEMBL6563725

CCOC(=O)C(OC)C1CCCN1C(=O)c1ccc(C#CCNc2ccc(C(=N)NC(=O)OC(C)(C)C)cc2)cc1C

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PTPN11 Q06124 1/20 0.33
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
DDB1 Q16531 1/20 0.31
CRBN Q96SW2 1/20 0.31
NPC1 O15118 1/20 0.31
ACACB O00763 1/20 0.30
JAK1 P23458 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565376 0.88 PRSS1 (0.35) GAASMN1; SMN2KMT2AALDH1A1ACACB
SCHEMBL6565417 0.86 PTPN11 (0.36) GAAPTPN11ALDH1A1HSP90AA1HSP90AB1
SCHEMBL6563779 0.86 KCNK3 (0.38) GAASMN1; SMN2PTPN11MEN1KMT2A
SCHEMBL7676439 0.84 HSD11B1 (0.32) GAASMN1; SMN2PTPN11MEN1KMT2A
SCHEMBL6565371 0.83 KCNK3 (0.34) GAASMN1; SMN2PTPN11MEN1KMT2A
SCHEMBL6565533 0.82 ACACB (0.45) GAAPTPN11MEN1KMT2AALDH1A1
SCHEMBL6565851 0.80 F2 (0.37) GAASMN1; SMN2ACACB
SCHEMBL6565336 0.80 ACACB (0.34) SMN1; SMN2PTPN11KMT2AALDH1A1NPC1
SCHEMBL6565215 0.79 PIK3CA (0.38) PTPN11DDB1CRBNACACBJAK1
SCHEMBL6561835 0.79 PTPN11 (0.35) GAAPTPN11MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed