SCHEMBL7808399

SCHEMBL7808399

CCOC(=O)c1ccccc1NCCCN1c2ccccc2CCc2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.51
CYP3A4 P08684 2/20 0.51
SLC6A2 P23975 2/20 0.51
SLC6A4 P31645 2/20 0.51
ADRA1A P35348 2/20 0.51
CYP1A2 P05177 2/20 0.51
CYP2D6 P10635 2/20 0.51
SLC22A2 O15244 1/20 0.51
SLC22A1 O15245 1/20 0.51
SLC22A3 O75751 1/20 0.51
CHRM2 P08172 1/20 0.51
CHRM1 P11229 1/20 0.51
DRD2 P14416 1/20 0.51
ADRA2B P18089 1/20 0.51
ADRA2C P18825 1/20 0.51
NFKB1 P19838 1/20 0.51
CHRM3 P20309 1/20 0.51
HTR2A P28223 1/20 0.51
HTR2C P28335 1/20 0.51
HRH1 P35367 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7810676 0.91 HDAC8 (0.55) MAPK1CYP3A4SLC6A2SLC6A4ADRA1A
SCHEMBL7604289 0.83 SLC6A2 (0.55) MAPK1CYP3A4SLC6A2SLC6A4ADRA1A
SCHEMBL9590321 0.78 TSHR (0.59) ADRA1AHTTKMT2ANPSR1KDM4E
SCHEMBL2296426 0.77 KDM4E (0.61) ADRA1AHTTKMT2ANPSR1KDM4E
SCHEMBL7808599 0.76 SLC6A4 (0.54) MAPK1CYP3A4SLC6A2SLC6A4ADRA1A
SCHEMBL7813757 0.76 SLC6A4 (0.54) MAPK1CYP3A4SLC6A2SLC6A4ADRA1A
SCHEMBL7634140 0.76 TSHR (0.56) MAPK1CYP3A4ADRA1AHTTKMT2A
SCHEMBL7609172 0.75 HDAC8 (0.61) MAPK1CYP3A4SLC6A2SLC6A4ADRA1A
Hydrochloric Acid SCHEMBL7813755 0.75 CYP3A4 (0.55) MAPK1CYP3A4SLC6A2SLC6A4ADRA1A
SCHEMBL11159593 0.75 TSHR (0.62) ADRA1AHTTKMT2ANPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820443-B1 HETEROCYCLIC COMPOUNDS FOR TREATING DIABETES NOVO NORDISK AS (DK) 2001-09-19 EP disclosed
EP-0820443-A1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1998-01-28 EP disclosed
WO-1996031481-A1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1996-10-10 WO disclosed