SCHEMBL7808442

SCHEMBL7808442

NC(c1ccccc1)c1ccc2[nH]c(CO)nc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
KDM4E B2RXH2 2/20 0.41
RAB9A P51151 2/20 0.41
GAA P10253 2/20 0.38
ALPL P05186 1/20 0.38
MAPK1 P28482 1/20 0.38
CHRM1 P11229 1/20 0.38
NPC1 O15118 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
DDAH1 O94760 1/20 0.36
POLB P06746 1/20 0.36
EGFR P00533 1/20 0.36
ERBB2 P04626 1/20 0.36
PKM P14618 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8478371 0.99 NPSR1 (0.44) TDP1NPSR1KDM4ERAB9AGAA
SCHEMBL7808444 0.89 TDP1 (0.52) TDP1NPSR1KDM4ERAB9AGAA
Hydrochloric Acid SCHEMBL8478379 0.88 NPSR1 (0.53) TDP1NPSR1KDM4ERAB9AGAA
SCHEMBL7806922 0.84 TDP1 (0.43) TDP1NPSR1KDM4ERAB9AGAA
Hydrochloric Acid SCHEMBL8480219 0.83 NPSR1 (0.45) TDP1NPSR1KDM4ERAB9AGAA
SCHEMBL8954822 0.75 CYP3A4 (0.48) TDP1KDM4ERAB9AMAPK1NPC1
SCHEMBL8954556 0.74 CHEK2 (0.37) NPSR1KDM4ERAB9ANPC1CYP1A2
SCHEMBL7806924 0.73 TDP1 (0.54) TDP1NPSR1KDM4ERAB9AGAA
Hydrochloric Acid SCHEMBL8955014 0.73 CHEK2 (0.36) NPSR1KDM4ERAB9ANPC1CYP1A2
SCHEMBL3947749 0.72 RAD52 (0.53) TDP1NPSR1KDM4ERAB9AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820990-B1 Benzimidazole, benzoxazole, and benzothiazole derivatives useful as interleukin 1beta inhibitors ADIR (FR) 2001-01-17 EP disclosed
EP-0820990-A2 Novel benzimidazole, benzoxazole, and benzothiazole derivatives useful as interleukin 1beta inhibitors ADIR ET COMPAGNIE (FR) 1998-01-28 EP disclosed