SCHEMBL7809114

SCHEMBL7809114

CCOC(=O)Cn1c(=O)c(=O)[nH]c2ccc(-n3ccnc3)cc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 3/20 0.49
GRIA2 P42262 3/20 0.49
GRIA3 P42263 3/20 0.49
GRIA4 P48058 3/20 0.49
SLC22A6 Q4U2R8 1/20 0.47
SLC22A8 Q8TCC7 1/20 0.47
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
MITF O75030 1/20 0.46
ALDH1A1 P00352 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
GRIK1 P39086 1/20 0.41
GRIK2 Q13002 1/20 0.41
GRIK3 Q13003 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8191168 0.84 SLC22A6 (0.56) GRIA1GRIA2GRIA3GRIA4SLC22A6
SCHEMBL8192729 0.82 SLC22A6 (0.55) GRIA1GRIA2GRIA3GRIA4SLC22A6
SCHEMBL8181436 0.82 SLC22A6 (0.55) GRIA1GRIA2GRIA3GRIA4SLC22A6
SCHEMBL8191992 0.82 SLC22A6 (0.55) GRIA1GRIA2GRIA3GRIA4SLC22A6
SCHEMBL8181377 0.82 SLC22A6 (0.54) GRIA1GRIA2GRIA3GRIA4SLC22A6
Hydrochloric Acid SCHEMBL8145152 0.81 PGR (0.43) SLC22A6SLC22A8PDE4APDE4BPDE4C
SCHEMBL8191185 0.81 SLC22A6 (0.53) GRIA1GRIA2GRIA3GRIA4SLC22A6
SCHEMBL7811473 0.80 SLC22A6 (0.52) GRIA1GRIA2GRIA3GRIA4SLC22A6
SCHEMBL8189778 0.80 GRIA1 (0.41) GRIA1GRIA2GRIA3GRIA4SLC22A6
SCHEMBL8191257 0.79 SLC22A6 (0.71) GRIA1GRIA2GRIA3GRIA4SLC22A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0784054-B1 1,2,3,4-TETRAHYDROQUINOXALINEDIONE DERIVATIVES AND USE AS GLUTAMATE RECEPTOR ANTAGONISTS YAMANOUCHI PHARMA CO LTD (JP) 2001-11-28 EP disclosed
CN-1067387-C 1,2,3,4-tetrahydroquinoxalindione derivative YAMANOUCHI PHARMA CO LTD (JP) 2001-06-20 CN disclosed
US-6096743-A 1,2,3,4-tetrahydroquinoxalinedione derivative YAMANOUCHI PHARMACEUTICALS CO., LTD. (JP) 2000-08-01 US disclosed
CN-1168670-A 1,2,3,4-tetrahydroquinoxalindione derivative YAMANOUCHI PHARMA CO LTD (JP) 1997-12-24 CN disclosed
EP-0784054-A1 1,2,3,4-TETRAHYDROQUINOXALINEDIONE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1997-07-16 EP disclosed