SCHEMBL7811149

SCHEMBL7811149

Clc1nsnc1C1CN2CCCC1C2

nearest known ligand 0.55

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 5/20 0.48
CHRM1 P11229 4/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7949366 1.00 CHRM2 (0.48) CHRM2CHRM1
SCHEMBL7949485 1.00 CHRM2 (0.48) CHRM2CHRM1
Hydrochloric Acid SCHEMBL7821090 0.98 CHRM2 (0.47) CHRM2CHRM1
Hydrochloric Acid SCHEMBL7949399 0.98 CHRM2 (0.47) CHRM2CHRM1
Oxalic Acid SCHEMBL7826358 0.93 CHRM2 (0.47) CHRM2CHRM1
SCHEMBL7818040 0.90 CHRM2 (0.46) CHRM2CHRM1
Oxalic Acid SCHEMBL7810405 0.85 CHRM2 (0.44) CHRM2CHRM1
SCHEMBL5931842 0.82 CHRM2 (0.44) CHRM2CHRM1
SCHEMBL13592143 0.81 CHRM2 (0.48) CHRM2CHRM1
SCHEMBL7810366 0.78 CHRM2 (0.56) CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 56 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0714394-B1 ANTIPSYCHOTIC METHOD WITH THIADIAZOLE AND OXADIAZOLE DERIVATIVES NOVO NORDISK AS (DK) 2001-06-20 EP claimed
EP-0866702-A1 METHOD FOR TREATING PAIN ELI LILLY AND COMPANY (US) 1998-09-30 EP claimed
WO-1997020556-A9 METHOD FOR TREATING PAIN 1997-10-02 WO claimed
WO-1997020556-A1 METHOD FOR TREATING PAIN ELI LILLY AND COMPANY (US) 1997-06-12 WO claimed
US-5574043-A ALZHEIMERS, GLAUCOMA, ANALGESIC NOVO NORDISK A/S (DK) 1996-11-12 US claimed
EP-0714394-A1 ANTIPSYCHOTIC METHOD NOVO NORDISK A/S (DK) 1996-06-05 EP claimed
WO-1996013168-A1 METHOD FOR TREATING ANXIETY ELI LILLY AND COMPANY (US) 1996-05-09 WO claimed
EP-0709095-A2 Method for treating anxiety using a tetrahydropyridine or azabicyclic oxadiazole or thiadiazole compound ELI LILLY AND COMPANY (US) 1996-05-01 EP claimed
WO-1995005379-A1 ANTIPSYCHOTIC METHOD NOVO NORDISK A/S (DK) 1995-02-23 WO claimed
EP-0544779-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1993-06-09 EP claimed
WO-1992003433-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1992-03-05 WO claimed
US-6281232-B1 AZABICYCLIC RING-SUBSTITUTED THIA- OR OXADIAZOLES NOVO NORDISK A/S (DK) 2001-08-28 US disclosed
US-6281233-B1 AZABICYCLIC RING-SUBSTITUTED THIA- OR OXADIAZOLES NOVO NORDISK A/S (DK) 2001-08-28 US disclosed
US-6271229-B1 ADMINISTERING A 1,2,5-OXADIAZOLE COMPOUND OR 1,2,5-THIADIAZOLE COMPOUND NOVO NORDISK A/S (DK) 2001-08-07 US disclosed
US-6265419-B1 IRRITABLE BOWEL DISORDER NOVO NORDISK A/S (DK) 2001-07-24 US disclosed
US-5260314-A Cognition activators, glaucoma analgesic NOVO NORDISK A/S (DK) 1993-11-09 US disclosed
WO-1993014089-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1993-07-22 WO disclosed
WO-1993014090-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1993-07-22 WO disclosed
EP-0544779-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1993-06-09 EP disclosed
WO-1992003433-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1992-03-05 WO disclosed