SCHEMBL7949366

SCHEMBL7949366

Clc1nsnc1[C@H]1CN2CCC[C@@H]1C2

nearest known ligand 0.55

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 5/20 0.48
CHRM1 P11229 4/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7811149 1.00 CHRM2 (0.48) CHRM2CHRM1
SCHEMBL7949485 1.00 CHRM2 (0.48) CHRM2CHRM1
Hydrochloric Acid SCHEMBL7821090 0.98 CHRM2 (0.47) CHRM2CHRM1
Hydrochloric Acid SCHEMBL7949399 0.98 CHRM2 (0.47) CHRM2CHRM1
Oxalic Acid SCHEMBL7826358 0.93 CHRM2 (0.47) CHRM2CHRM1
SCHEMBL7818040 0.90 CHRM2 (0.46) CHRM2CHRM1
Oxalic Acid SCHEMBL7810405 0.85 CHRM2 (0.44) CHRM2CHRM1
SCHEMBL5931842 0.82 CHRM2 (0.44) CHRM2CHRM1
SCHEMBL13592143 0.81 CHRM2 (0.48) CHRM2CHRM1
SCHEMBL7810366 0.78 CHRM2 (0.56) CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6271229-B1 ADMINISTERING A 1,2,5-OXADIAZOLE COMPOUND OR 1,2,5-THIADIAZOLE COMPOUND NOVO NORDISK A/S (DK) 2001-08-07 US claimed
WO-1996014316-A1 A METHOD OF TREATING URINARY BLADDER DYSFUNCTIONS NOVO NORDISK A/S (DK) 1996-05-17 WO claimed
US-6281232-B1 AZABICYCLIC RING-SUBSTITUTED THIA- OR OXADIAZOLES NOVO NORDISK A/S (DK) 2001-08-28 US disclosed
US-6281233-B1 AZABICYCLIC RING-SUBSTITUTED THIA- OR OXADIAZOLES NOVO NORDISK A/S (DK) 2001-08-28 US disclosed
US-6271229-B1 ADMINISTERING A 1,2,5-OXADIAZOLE COMPOUND OR 1,2,5-THIADIAZOLE COMPOUND NOVO NORDISK A/S (DK) 2001-08-07 US disclosed
US-6265419-B1 IRRITABLE BOWEL DISORDER NOVO NORDISK A/S (DK) 2001-07-24 US disclosed
US-5612351-A AZABICYCLIC DERIVATIVES OF 1,2,3-OXA(OR THIA)DIAZOLE NOVO NORDISK A/S (DK) 1997-03-18 US disclosed
WO-1996014316-A1 A METHOD OF TREATING URINARY BLADDER DYSFUNCTIONS NOVO NORDISK A/S (DK) 1996-05-17 WO disclosed