SCHEMBL7811348

SCHEMBL7811348

COc1cccc(CN(C)C(=O)CC(CCO)c2ccc(Cl)c(Cl)c2)c1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.47
HSD17B2 P37059 4/20 0.43
TDP1 Q9NUW8 1/20 0.43
TSPO P30536 5/20 0.43
DPP4 P27487 1/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
POLB P06746 1/20 0.41
HPGD P15428 1/20 0.41
RECQL P46063 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7802828 0.91 TACR1 (0.56) TACR1TDP1SMN1; SMN2
SCHEMBL7809340 0.89 TACR1 (0.51) TACR1HSD17B2TDP1TSPOMEN1
SCHEMBL7809517 0.87 TACR1 (0.47) TACR1HSD17B2TDP1TSPODPP4
SCHEMBL7815209 0.86 TACR1 (0.50) TACR1TDP1MEN1KMT2AHPGD
SCHEMBL7807768 0.85 TACR1 (0.44) TACR1HSD17B2TDP1TSPODPP4
SCHEMBL7807544 0.82 KDM4E (0.45) TDP1
SCHEMBL6973685 0.81 MEN1 (0.47) TACR1TDP1MEN1KMT2ABCHE
SCHEMBL7811515 0.81 ALDH1A1 (0.55) TACR1BCHESMN1; SMN2POLBHPGD
SCHEMBL7815520 0.79 TACR1 (0.60) TACR1TDP1SMN1; SMN2
SCHEMBL7815376 0.78 FFAR1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773929-B1 PIPERIDINE DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORP (US) 2001-10-31 EP disclosed
US-5654316-A Piperidine derivatives as neurokinin antagonists SCHERING CORPORATION (US) 1997-08-05 US disclosed