SCHEMBL7813239

SCHEMBL7813239

CC(C)(C)[Si](OCc1ccc(C(O)=S)cc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PPARG P37231 3/20 0.36
RXRA P19793 4/20 0.36
RXRB P28702 3/20 0.36
RXRG P48443 2/20 0.36
SMYD2 Q9NRG4 2/20 0.33
PPARA Q07869 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
NR4A2 P43354 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ATM Q13315 1/20 0.32
MAOB P27338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9342265 0.85 RXRA (0.51) PPARGRXRARXRBRXRGNR4A2
SCHEMBL9347235 0.84 ESR1 (0.43) PPARGALDH1A1ATM
SCHEMBL1314001 0.84 AGXT (0.42) SMYD2ALDH1A1HTTSMN1; SMN2L3MBTL1
SCHEMBL5918964 0.84 MAOB (0.50) PPARGRXRARXRBRXRGALDH1A1
SCHEMBL2745018 0.83 PPARG (0.41) PPARGRXRARXRBRXRGPPARA
SCHEMBL14542685 0.81 AGXT (0.43) CA1CA2CA9ALDH1A1HTT
SCHEMBL11934179 0.81 TP53 (0.42) PPARGRXRARXRBSMYD2PPARA
SCHEMBL9347236 0.80 AGXT (0.33) PPARGRXRARXRBRXRGSMYD2
SCHEMBL4587307 0.80 IDO1 (0.42) HTTSMN1; SMN2L3MBTL1MAOB
SCHEMBL222047 0.80 MAOB (0.43) SMN1; SMN2L3MBTL1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0574784-B1 Process for preparing (1'R,3S,4R)4-acylthio azetidinones PHARMACIA & UPJOHN SPA (IT) 2001-12-05 EP disclosed
US-5399679-A (1'R,3S,4R)4-acylthio azetidinones FARMITALIA CARLO ERBA S.R.L. (IT) 1995-03-21 US disclosed
WO-1993025523-A1 4-ACYLTHIO AZETIDINONES FARMITALIA CARLO ERBA S.R.L. (IT) 1993-12-23 WO disclosed
EP-0574784-A1 (1'R,3S,4R)4-acylthio azetidinones PHARMACIA S.p.A. (IT) 1993-12-22 EP disclosed