SCHEMBL78163

SCHEMBL78163

COc1cc(COc2cccc(C(C)(C)C)c2)cc(OC)c1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOB P27338 9/20 0.57
APP P05067 1/20 0.53
SOD1 P00441 1/20 0.52
ABCB1 P08183 1/20 0.48
NR4A1 P22736 1/20 0.48
NR4A2 P43354 1/20 0.48
NR4A3 Q92570 1/20 0.48
MRGPRX4 Q96LA9 1/20 0.47
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.45
HTT P42858 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
BCHE P06276 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13439849 0.91 MAOB (0.61) MAOBAPPSOD1ABCB1MRGPRX4
SCHEMBL13439834 0.88 NPC1 (0.58) MAOBAPPSOD1NR4A1NR4A2
SCHEMBL791326 0.83 MAOB (0.69) MAOBAPPNR4A1NR4A2NR4A3
SCHEMBL78171 0.82 MAOB (0.62) MAOBSOD1NR4A1NR4A2NR4A3
SCHEMBL7917111 0.82 MAOB (0.62) MAOBAPPABCB1MRGPRX4NPC1
SCHEMBL29303965 0.82 APP (0.58) MAOBAPPNR4A2LMNAPOLB
SCHEMBL22548672 0.79 MAOB (0.56) MAOBNR4A2MRGPRX4LMNAHTT
SCHEMBL13761594 0.79 NR4A2 (0.56) MAOBAPPSOD1NR4A1NR4A2
SCHEMBL146154 0.79 ACHE (0.52) SOD1LMNAPOLBHTTL3MBTL1
SCHEMBL5987976 0.79 MAOB (0.76) MAOBAPPABCB1MRGPRX4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed