SCHEMBL7817697

SCHEMBL7817697

O=C(NCCCCN1CCN(c2csc3cc(F)ccc23)CC1)c1ccc(F)cc1

nearest known ligand 0.73

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 4/20 0.73
DRD2 P14416 10/20 0.60
DRD3 P35462 9/20 0.60
DRD4 P21917 8/20 0.60
HTR1A P08908 7/20 0.60
ADRA1D P25100 2/20 0.60
ADRA1B P35368 2/20 0.60
HTR2A P28223 5/20 0.54
HTR2C P28335 3/20 0.51
HTR2B P41595 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13809546 0.94 ADRA1A (0.69) ADRA1ADRD2DRD3DRD4HTR1A
SCHEMBL13809559 0.94 ADRA1A (0.69) ADRA1ADRD2DRD3DRD4HTR1A
SCHEMBL13809551 0.94 ADRA1A (0.68) ADRA1ADRD2DRD3DRD4HTR1A
SCHEMBL13809541 0.93 ADRA1A (0.67) ADRA1ADRD2DRD3DRD4HTR1A
SCHEMBL13809533 0.90 ADRA1A (0.66) ADRA1ADRD2DRD3DRD4HTR1A
SCHEMBL13809537 0.90 ADRA1A (0.65) ADRA1ADRD2DRD3DRD4HTR1A
SCHEMBL13809557 0.89 ADRA1A (0.64) ADRA1ADRD2DRD3DRD4HTR1A
SCHEMBL13809566 0.89 ADRA1A (0.71) ADRA1ADRD2DRD3DRD4HTR1A
SCHEMBL7824411 0.88 ADRA1A (0.70) ADRA1ADRD2DRD3DRD4HTR1A
SCHEMBL13809562 0.88 ADRA1A (0.70) ADRA1ADRD2DRD3DRD4HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0732332-A1 Substituted benzothienylpiperazines, their use as medicaments, and processes for their preparation HOECHST MARION ROUSSEL, INC. (US) 1996-09-18 EP claimed
EP-0732332-B1 Substituted benzothienylpiperazines, their use as medicaments, and processes for their preparation AVENTIS PHARMA INC (US) 2001-12-19 EP disclosed
EP-0732332-A1 Substituted benzothienylpiperazines, their use as medicaments, and processes for their preparation HOECHST MARION ROUSSEL, INC. (US) 1996-09-18 EP disclosed