SCHEMBL7818489

SCHEMBL7818489

Cc1cccc2c1C(C)NCC2

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.42
DRD2 P14416 3/20 0.42
PARP1 P09874 1/20 0.41
PRCP P42785 3/20 0.40
MAOA P21397 3/20 0.40
DRD3 P35462 2/20 0.40
TSHR P16473 2/20 0.40
KDM4E B2RXH2 1/20 0.40
CYP2C9 P11712 1/20 0.40
HIF1A Q16665 1/20 0.40
HSD17B10 Q99714 1/20 0.40
DRD4 P21917 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19684816 1.00 HTR2C (0.42) HTR2CDRD2PARP1PRCPMAOA
SCHEMBL19684822 1.00 HTR2C (0.42) HTR2CDRD2PARP1PRCPMAOA
SCHEMBL19711049 0.80 HTR2C (0.41) HTR2CDRD2PARP1PRCPMAOA
SCHEMBL1010276 0.80 HTR2C (0.41) HTR2CDRD2PARP1PRCPMAOA
SCHEMBL30983663 0.80 HTR2C (0.41) HTR2CDRD2PARP1PRCPMAOA
SCHEMBL19711053 0.80 HTR2C (0.41) HTR2CDRD2PARP1PRCPMAOA
SCHEMBL19678842 0.77 PARP1 (0.41) HTR2CDRD2PARP1PRCPMAOA
SCHEMBL19678841 0.77 PARP1 (0.41) HTR2CDRD2PARP1PRCPMAOA
SCHEMBL12311985 0.77 MAOA (0.53) HTR2CDRD2MAOATSHRHSD17B10
SCHEMBL21651084 0.77 PRCP (0.57) DRD2PRCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3464249-B1 SUBSTITUTED CARBONUCLEOSIDE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER (US) 2021-08-11 EP disclosed
EP-0677049-B1 QUINAZOLINE DERIVATIVES YUHAN CORP LTD (KR) 2001-07-25 EP disclosed
US-5686458-A Quinazoline deriviates for treating peptic ulcer YUHAN CORPORATION (KR) 1997-11-11 US disclosed
EP-0677049-A1 QUINAZOLINE DERIVATIVES YUHAN CORPORATION, LTD. (KR) 1995-10-18 EP disclosed
WO-1994014795-A1 QUINAZOLINE DERIVATIVES YUHAN CORPORATION (KR) 1994-07-07 WO disclosed