SCHEMBL7821768

SCHEMBL7821768

N#CC(=Cc1cccc(O)c1)C(=O)OC(C(=O)O)c1ccc(F)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.56
MAPT P10636 4/20 0.48
KMT2A Q03164 3/20 0.46
MEN1 O00255 1/20 0.46
EGFR P00533 1/20 0.42
ERBB2 P04626 1/20 0.42
ALDH1A1 P00352 4/20 0.41
PDCD1 Q15116 1/20 0.41
CD274 Q9NZQ7 1/20 0.41
LMNA P02545 2/20 0.40
MAPK1 P28482 1/20 0.40
TDP1 Q9NUW8 2/20 0.40
RECQL P46063 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
DNM1 Q05193 2/20 0.39
MMP1 P03956 1/20 0.38
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
POLB P06746 1/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Alpha-Cyano-3-Hydroxycinnamic Acid SCHEMBL7821767 0.81 KDM4E (0.68) KDM4EMAPTKMT2AMEN1EGFR
SCHEMBL7821773 0.80 KDM4E (0.53) KDM4EMAPTKMT2AMEN1EGFR
SCHEMBL21457685 0.77 KDM4E (0.65) KDM4EMAPTKMT2AMEN1ALDH1A1
SCHEMBL21457688 0.77 KDM4E (0.65) KDM4EMAPTKMT2AMEN1ALDH1A1
Alpha-Cyano-3-Hydroxycinnamic Acid SCHEMBL1285559 0.73 KDM4E (1.00) KDM4EMAPTKMT2AMEN1EGFR
Alpha-Cyano-3-Hydroxycinnamic Acid SCHEMBL2057244 0.73 KDM4E (1.00) KDM4EMAPTKMT2AMEN1EGFR
Alpha-Cyano-3-Hydroxycinnamic Acid SCHEMBL29881895 0.73 KDM4E (1.00) KDM4EMAPTKMT2AMEN1EGFR
Alpha-Cyano-3-Hydroxycinnamic Acid SCHEMBL1285555 0.73 KDM4E (1.00) KDM4EMAPTKMT2AMEN1EGFR
SCHEMBL21457224 0.73 KDM4E (0.70) KDM4EMAPTKMT2AMEN1EGFR
SCHEMBL21457227 0.73 KDM4E (0.70) KDM4EMAPTKMT2AMEN1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091958-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2001-04-18 EP disclosed
WO-2000001692-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2000-01-13 WO disclosed