SCHEMBL7821787

SCHEMBL7821787

O=CN(C=O)CC(=O)c1ccccc1C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.52
ALOX15 P16050 1/20 0.52
AKR1C3 P42330 1/20 0.42
USP2 O75604 1/20 0.41
TP53 P04637 1/20 0.41
KDM4E B2RXH2 2/20 0.41
HMGB1 P09429 2/20 0.41
HPGD P15428 2/20 0.41
NAPRT Q6XQN6 2/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA6 P23280 1/20 0.41
CA7 P43166 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
KMT2A Q03164 2/20 0.40
APEX1 P27695 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10028289 0.80 TSHR (0.47) ALDH1A1ALOX15KDM4ECA1CA2
SCHEMBL8015832 0.77 TSHR (0.64) ALDH1A1TP53KDM4ETDP1L3MBTL1
SCHEMBL8227137 0.77 CTNNB1 (0.53) ALDH1A1TP53KDM4EHPGDSMN1; SMN2
SCHEMBL2818404 0.76 NPC1 (0.54) ALDH1A1TP53HPGDSMN1; SMN2KMT2A
Phthalic Acid SCHEMBL28415888 0.74 ALDH1A1 (0.93) ALDH1A1ALOX15AKR1C3KDM4EHMGB1
Phthalic Acid SCHEMBL198844 0.74 ALDH1A1 (0.93) ALDH1A1ALOX15AKR1C3KDM4EHMGB1
SCHEMBL11950516 0.73 ALDH1A1 (0.70) ALDH1A1ALOX15AKR1C3USP2TP53
Phthalic Acid SCHEMBL5903044 0.73 ALDH1A1 (0.78) ALDH1A1ALOX15AKR1C3KDM4EHMGB1
Phthalic Acid SCHEMBL29285423 0.73 ALDH1A1 (0.78) ALDH1A1ALOX15AKR1C3KDM4EHMGB1
Phthalic Acid SCHEMBL10731126 0.72 ALDH1A1 (0.88) ALDH1A1ALOX15AKR1C3KDM4EHMGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880522-B1 5H,10H-IMIDAZO[1,2-a]INDENO[1,2-e]PYRAZINE-4-ONE DERIVATIVES AMPA AND NMDA RECEPTORS ANTAGONISTS, PREPARATION THEREOF, INTERMEDIATES THEREOF AND DRUGS CONTAINING SAME AVENTIS PHARMA SA (FR) 2001-09-19 EP disclosed
EP-0880522-A1 5H,10H-IMIDAZO 1,2-a]INDENO 1,2-e]PYRAZINE-4-ONE DERIVATIVES, PREPARATION THEREOF, INTERMEDIATES THEREOF AND DRUGS CONTAINING SAME Aventis Pharma S.A. (FR) 1998-12-02 EP disclosed
WO-1997025328-A1 5H,10H-IMIDAZO[1,2-a]INDENO[1,2-e]PYRAZINE-4-ONE DERIVATIVES, PREPARATION THEREOF, INTERMEDIATES THEREOF AND DRUGS CONTAINING SAME RHONE-POULENC RORER S.A. (FR) 1997-07-17 WO disclosed