SCHEMBL7821841

SCHEMBL7821841

O=S(=O)(Cc1ccccc1)N1CCc2ccccc2C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.59
MEN1 O00255 5/20 0.59
ALDH1A1 P00352 3/20 0.59
TSHR P16473 2/20 0.59
POLB P06746 1/20 0.59
MAPT P10636 1/20 0.59
HPGD P15428 1/20 0.58
RORC P51449 2/20 0.50
AKR1C3 P42330 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30539315 1.00 KMT2A (0.59) KMT2AMEN1ALDH1A1TSHRPOLB
SCHEMBL31670446 0.84 AKR1C3 (0.53) KMT2AMEN1ALDH1A1TSHRPOLB
SCHEMBL6393137 0.84 TSHR (0.49) KMT2AMEN1ALDH1A1TSHRPOLB
SCHEMBL17227611 0.83 KMT2A (0.62) KMT2AMEN1TSHRPOLBMAPT
SCHEMBL3282591 0.82 AKR1C3 (0.53) TSHRHPGDRORCAKR1C3
SCHEMBL6398959 0.80 AKR1C3 (0.56) KMT2AMEN1ALDH1A1TSHRPOLB
SCHEMBL23657779 0.79 KMT2A (0.50) KMT2AMEN1ALDH1A1TSHRHPGD
SCHEMBL5069905 0.79 TSHR (0.49) KMT2AMEN1ALDH1A1TSHRPOLB
SCHEMBL7076783 0.79 AKR1C3 (0.52) KMT2AMEN1ALDH1A1TSHRPOLB
SCHEMBL735675 0.79 TSHR (0.81) KMT2AALDH1A1TSHRPOLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140834-A1 HETEROCYCLIC PIPERIDINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Du Pont Pharmaceuticals Company (US) 2001-10-10 EP claimed
WO-2000035877-A1 HETEROCYCLIC PIPERIDINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY DU PONT PHARMACEUTICALS COMPANY (US) 2000-06-22 WO claimed
EP-1140834-A1 HETEROCYCLIC PIPERIDINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Du Pont Pharmaceuticals Company (US) 2001-10-10 EP disclosed
WO-2000035877-A1 HETEROCYCLIC PIPERIDINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY DU PONT PHARMACEUTICALS COMPANY (US) 2000-06-22 WO disclosed