SCHEMBL7824031

SCHEMBL7824031

O=Cc1c[nH]c2ccc(CCC(Br)I)cc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C19 P33261 1/20 0.46
CYP2A6 P11509 3/20 0.43
IMPDH2 P12268 1/20 0.43
CCNT1 O60563 1/20 0.37
CDK9 P50750 1/20 0.37
HASPIN Q8TF76 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
PIM3 Q86V86 2/20 0.36
PIM1 P11309 1/20 0.36
GABRP O00591 2/20 0.36
GABRD O14764 2/20 0.36
GABRA1 P14867 2/20 0.36
GABRB1 P18505 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7834310 0.83 ALDH1A1 (0.48) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL7823204 0.79 ALDH1A1 (0.50) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL7229792 0.79 ALDH1A1 (0.51) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL7823270 0.78 CYP2A6 (0.42) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL5814027 0.78 ALDH1A1 (0.54) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL13592398 0.78 ALDH1A1 (0.54) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL8746106 0.77 CYP2A6 (0.56) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL5403384 0.75 ALDH1A1 (0.58) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL7856276 0.74 ALDH1A1 (0.61) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2
SCHEMBL7837902 0.74 ALDH1A1 (0.50) ALDH1A1CYP1A2CYP2C19CYP2A6IMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1109813-A1 PYRROLOINDOLES, PYRIDOINDOLES AND AZEPINOINDOLES AS 5-HT2C AGONISTS VERNALIS RESEARCH LIMITED (GB) 2001-06-27 EP disclosed
WO-2000012510-A1 PYRROLOINDOLES, PYRIDOINDOLES AND AZEPINOINDOLES AS 5-HT2C AGONISTS VERNALIS RESEARCH LIMITED (GB) 2000-03-09 WO disclosed