SCHEMBL7825490

SCHEMBL7825490

CC(=O)c1c(OC(C)C(=O)O)ccc2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NCEH1 Q6PIU2 4/20 0.56
PPARG P37231 4/20 0.50
PPARA Q07869 4/20 0.50
KMT2A Q03164 2/20 0.50
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
GAA P10253 1/20 0.43
PKM P14618 1/20 0.43
MAPT P10636 2/20 0.42
TSHR P16473 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
APEX1 P27695 1/20 0.41
CTSD P07339 1/20 0.41
AKR1B1 P15121 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16329074 0.86 NCEH1 (0.60) NCEH1CYP1A2CYP2C9CYP2C19MAPT
SCHEMBL27945004 0.82 KMT2A (0.53) NCEH1PPARGPPARAKMT2ACYP1A2
SCHEMBL2922977 0.80 PPARG (0.64) PPARGPPARAKMT2ACYP1A2CYP2C9
SCHEMBL16933412 0.80 PPARG (0.64) PPARGPPARAKMT2ACYP1A2CYP2C9
SCHEMBL31376342 0.80 PPARG (0.64) PPARGPPARAKMT2ACYP1A2CYP2C9
SCHEMBL16933413 0.80 PPARG (0.64) PPARGPPARAKMT2ACYP1A2CYP2C9
SCHEMBL2563368 0.78 CYP1A2 (0.71) NCEH1PPARGPPARAKMT2ACYP1A2
SCHEMBL3357585 0.78 NCEH1 (0.65) NCEH1KMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL30676839 0.78 NCEH1 (0.65) NCEH1KMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL28423314 0.77 CYP1A2 (0.56) NCEH1KMT2ACYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1131288-A1 PYRROLIDINE DERIVATIVES-CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-09-12 EP disclosed
EP-1091958-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2001-04-18 EP disclosed
US-6166015-A Pyrrolidine derivatives-CCR-3 receptor antagonists SYNTEX (U.S.A.) INC. (US) 2000-12-26 US disclosed
WO-2000031032-A1 PYRROLIDINE DERIVATIVES-CCR-3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-02 WO disclosed
WO-2000001692-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2000-01-13 WO disclosed