SCHEMBL7825901

SCHEMBL7825901

CN1CCN(C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)[C@H](Cc2cn(C)c3ccccc23)C1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 18/20 0.51
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA4 P22748 2/20 0.44
CA9 Q16790 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8480574 1.00 TACR1 (0.51) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL8478985 0.99 TACR1 (0.50) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL7815938 0.99 TACR1 (0.50) TACR1CA1CA2CA4CA9
SCHEMBL7829861 0.90 TACR1 (0.49) TACR1CA1CA2CA4CA9
SCHEMBL7826647 0.88 TACR1 (0.51) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL7830176 0.87 TACR1 (0.51) TACR1CA1CA2CA4CA9
SCHEMBL7650068 0.86 TACR1 (0.47) TACR1
SCHEMBL8478086 0.85 IDE (0.49) TACR1CA1CA2CA4CA9
SCHEMBL7122736 0.85 IDE (0.49) TACR1CA1CA2CA4CA9
Hydrochloric Acid SCHEMBL8475499 0.81 TACR1 (0.64) TACR1CA1CA2CA4CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655442-B1 Piperazine derivatives as Tachykinin antagonists FUJISAWA PHARMACEUTICAL CO (JP) 2001-05-23 EP disclosed
EP-0655442-A1 Piperazine derivatives as Tachykinin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-05-31 EP disclosed